Clinical trial • Phase III • Neurology|Rare Disease

Allopurinol sodium for Hypoxic-ischemic encephalopathy (HIE)|Neonatal asphyxia

Phase III trial of Allopurinol sodium for Hypoxic-ischemic encephalopathy (HIE)|Neonatal asphyxia.

Overview

Trial Therapeutic Area
Neurology|Rare Disease
Trial Disease
Hypoxic-ischemic encephalopathy (HIE)|Neonatal asphyxia
Trial Stage
Phase III
Drug Modality
Small molecule
Paediatric Trial
Yes
Orphan Drug
Yes

Key dates

Initial CTIS Submission Date
06-08-2024
First CTIS Authorization Date
10-09-2024

Trial design

Randomised, placebo arm: mannitol (solution for infusion) administered iv as placebo; allopurinol (acepurin) investigational arm administered iv (active substance: allopurinol sodium). dosing unit information present (mg/kg) with max daily dose amount 30 mg/kg; study is placebo-controlled and compares allopurinol plus standard of care versus placebo plus standard of care (standard care may include therapeutic hypothermia if indicated). Phase III trial across 36 sites in Germany, Italy, Norway and others.

Randomised
Yes
Comparator
Placebo arm: MANNITOL (solution for infusion) administered IV as placebo; Allopurinol (ACEPURIN) investigational arm administered IV (active substance: allopurinol sodium). Dosing unit information present (mg/kg) with max daily dose amount 30 mg/kg; study is placebo-controlled and compares allopurinol plus standard of care versus placebo plus standard of care (standard care may include therapeutic hypothermia if indicated).
Trial Duration For Participant
730

Eligibility

Recruits 452 paediatric patients.

Vulnerable Population
Neonates (newborns) are a vulnerable population; consent is obtained from parents/legal guardians. Subject information and informed consent forms for parents/guardians are provided (country-specific documents listed in multiple languages). Assent is not applicable for neonates.

Inclusion criteria

  • {"criterion_text":"- Severe perinatal metabolic acidosis or ongoing cardiopulmonary resuscitation at 5 min after birth\n- Early clinical signs of potentially evolving encephalopathy"}

Exclusion criteria

  • {"criterion_text":"- gestational age below 36 weeks\n- birth weight below 2500 g\n- postnatal age >30min at the end of screening phase\n- severe congenital malformation or syndrome requiring neonatal surgery or affecting long-term outcome\n- patient considered “moribund” / “non-viable” (e.g., lack of spontaneous cardiac activity and ongoing chest compression at 30min)"}

Endpoints

Primary endpoints

  • {"endpoint_text":"- Death versus severe neurodevelopmental impairment versus survival without severe neurodevelopmental impairment at the age of two years","definition_or_measurement_approach":"Severe neurodevelopmental impairment defined as cerebral palsy, or cognitive or language impairment (cognitive- and language-composite scores of the Bayley Scales of Infant and Toddler Development, 3rd edition <85) assessed at 24 months of age."}

Secondary endpoints

  • {"endpoint_text":"- Death or neurodevelopmental impairment (NDI) The primary endpoint will be reconstituted as dichotomised composite secondary endpoint (survival without NDI versus Death or languagecomposite- score < 85 or cognitive-composite-score <85 or cerebral palsy present).","definition_or_measurement_approach":"Dichotomised composite: survival without NDI versus death or Bayley language-composite <85 or cognitive-composite <85 or presence of cerebral palsy."}
  • {"endpoint_text":"- Incidence of CP Incidence of CP will be analyzed by Cochrane-Mantel-Haenzel- X²-Test.","definition_or_measurement_approach":"Incidence of cerebral palsy analyzed using Cochrane-Mantel-Haenszel chi-square test."}
  • {"endpoint_text":"- GMFCS-score GMFCS-Score for quantification of the effects of cerebral palsy and other motor impairments (adapted from Palisano et al. [Palisano Med Child Neurol 1997]) using the ALBINO-GMFCS-score sheet (separate document not part of this protocol) will be analysed. GMFCS-score consists of six categories.","definition_or_measurement_approach":"Gross Motor Function Classification System (GMFCS) categories (six categories) assessed using ALBINO-GMFCS-score sheet."}
  • {"endpoint_text":"- Motor-Composite-Score (Bayley III)","definition_or_measurement_approach":"Motor composite score from Bayley Scales of Infant and Toddler Development, 3rd edition."}
  • {"endpoint_text":"- Motor-Composite-Score dichotomised (Bayley III) The motor-composite-score will be dichotomised at the cut-off <85 versus ≥85","definition_or_measurement_approach":"Motor-composite score dichotomised at <85 versus ≥85."}
  • {"endpoint_text":"- Cognitive-Composite-Score (cognitive subscale, Bayley III)","definition_or_measurement_approach":"Cognitive composite score from Bayley III cognitive subscale."}
  • {"endpoint_text":"- Cognitive-Composite-Score dichotomised (cognitive subscale, Bayley III) The cognitive-composite-score will be dichotomised at the cut-off <85 versus ≥85","definition_or_measurement_approach":"Cognitive-composite score dichotomised at <85 versus ≥85."}
  • {"endpoint_text":"- Language-Composite-Score (language subscale, Bayley III)","definition_or_measurement_approach":"Language composite score from Bayley III language subscale."}
  • {"endpoint_text":"- Language-Composite-Score dichotomised (language subscale, Bayley III) The language-composite-score will be dichotomised at the cut-off <85 versus ≥85","definition_or_measurement_approach":"Language-composite score dichotomised at <85 versus ≥85."}
  • {"endpoint_text":"- Single Components of primary endpoint - Graph Single components and observed combinations of the primary endpoint (healthy, death, CP, language-composite-score <85, cognitive-composite- score <85) will be displayed graphically stratified for the two treatment groups.","definition_or_measurement_approach":"Graphical display of individual components and observed combinations of primary endpoint stratified by treatment group."}

Recruitment

Recruitment Window Months
99
Consent Approach
Informed consent is provided by parents/legal guardians (parents and guardians ICFs available). Subject information and informed consent forms for parents/guardians are provided as country-specific documents; available languages/country documents include (examples in documents list) English, Dutch, German, French, Spanish, Finnish, Russian, Italian and country-specific translations. Assent is not applicable for neonates.

Geography

Total Number Of Sites
36
Total Number Of Participants
452

Germany

Earliest CTIS Part Ii Submission Date
22-08-2024
Latest Decision Or Authorization Date
14-01-2025
Processing Time Days
145
Number Of Sites
8
Number Of Participants
112

Sites

Site Name
Universitaetsklinikum Muenster AöR
Department Name
Neonatology
Contact Person Name
Jenny Potratz
Contact Person Email
jenny.potratz@ukmuenster.de
Site Name
Universitaet Leipzig
Department Name
Neonatology
Contact Person Name
Ulrich Thome
Site Name
Universitaetsklinikum Duesseldorf AöR
Department Name
Neonatology
Contact Person Name
Thomas Hoehn
Site Name
Cnopf'sche Kinderklinik/Klinik Hallerwiese
Department Name
Neonatology
Contact Person Name
Michael Schroth
Contact Person Email
michael.schroth@diakoneo.de
Site Name
Auf der Bult Kinder- und Jugendkrankenhaus
Department Name
Neonatology
Contact Person Name
Anna Koluch
Contact Person Email
koluch@hka.de
Site Name
University Of Tuebingen
Department Name
Neonatology
Contact Person Name
Axel Franz
Site Name
KJF Klinik Josefinum, Klinik für Kinder und Jugendliche
Department Name
Neonatology
Contact Person Name
Thomas Völkl
Contact Person Email
voelkl.thomas@josefinum.de
Site Name
Universitaetsklinikum Carl Gustav Carus Dresden an der Technischen Universitaet Dresden AöR
Department Name
Neonatology
Contact Person Name
Barbara Seipolt

Italy

Earliest CTIS Part Ii Submission Date
22-08-2024
Latest Decision Or Authorization Date
20-05-2025
Processing Time Days
271
Number Of Sites
3
Number Of Participants
23

Sites

Site Name
ASST FBF-Sacco Ospedale dei Bambini "V.Buzzi"
Department Name
Neonatology
Contact Person Name
Gianluca Lista
Site Name
Azienda Sanitaria Universitaria Friuli Centrale (ASUFC)
Department Name
Neonatology
Contact Person Name
Isabella Mauro
Site Name
Azienda Ospedaliero Universitaria Ospedali Riuniti Umberto I G M Lancisi G Salesi
Department Name
Neonatology
Contact Person Name
Virgilio Carnielli
Contact Person Email
v.carnielli@staff.univpm.it

Norway

Earliest CTIS Part Ii Submission Date
22-08-2024
Latest Decision Or Authorization Date
10-09-2024
Processing Time Days
19
Number Of Sites
1
Number Of Participants
36

Sites

Site Name
Oslo Universitetssykehus UUS
Department Name
Neonatology
Contact Person Name
Mari Falck
Contact Person Email
mfalck@ous-hf.no

Spain

Earliest CTIS Part Ii Submission Date
22-08-2024
Latest Decision Or Authorization Date
06-08-2025
Processing Time Days
349
Number Of Sites
2
Number Of Participants
32

Sites

Site Name
Hospital Universitario La Fe
Department Name
Neonatology
Contact Person Name
Maximo Vento
Contact Person Email
maximo.vento@uv.es
Site Name
Hospital General Alicante
Department Name
Neonatology
Contact Person Name
Caridad Tapia Collados
Contact Person Email
ctapiac@coma.es

Finland

Earliest CTIS Part Ii Submission Date
22-08-2024
Latest Decision Or Authorization Date
12-09-2024
Processing Time Days
21
Number Of Sites
2
Number Of Participants
67

Sites

Site Name
Helsingin ja Uudenmaan Sairaanhoitopiirin Kuntayhtämy (HUS)
Department Name
Neonatology
Contact Person Name
Marjo Metsäranta
Contact Person Email
marjo.metsaranta@hus.fi
Site Name
Jorvi Hospital, HUS
Department Name
Neonatology
Contact Person Name
Marjo Metsäranta
Contact Person Email
marjo.metsaranta@hus.fi

Netherlands

Earliest CTIS Part Ii Submission Date
22-08-2024
Latest Decision Or Authorization Date
06-08-2025
Processing Time Days
349
Number Of Sites
13
Number Of Participants
90

Sites

Site Name
St. Antonius Ziekenhuis
Department Name
Neonatology
Contact Person Name
Jacqueline van Hillegersberg
Site Name
Deventer Ziekenhuis
Department Name
Neonatology
Contact Person Name
Anne Dassel
Contact Person Email
c.dassel@dz.nl
Site Name
Maxima Medisch Centrum
Department Name
Neonatology
Contact Person Name
Koenraad Dijkman
Contact Person Email
k.dijkman@mmc.nl
Site Name
Universitair Medisch Centrum Utrecht
Department Name
Neonatology
Contact Person Name
Frank van Bel
Contact Person Email
f.vanbel@umcutrecht.nl
Site Name
Isala Kliniek Zwolle
Department Name
Neonatology
Contact Person Name
Marianne van der Heide
Contact Person Email
m.jalving@isala.nl
Site Name
Diakonessenhuis Stichting
Department Name
Neonatology
Contact Person Name
Inge de Boer
Contact Person Email
idboer@diakhuis.nl
Site Name
Sint Elisabeth Ziekenhuis Tilburg
Department Name
Neonatology
Contact Person Name
Carien Smeets
Contact Person Email
c.smeets@elisabeth.nl
Site Name
Spaarne Gasthuis
Department Name
Neonatology
Contact Person Name
Marianne van Houten
Site Name
Vumc Medical Center - Emma's Children's Hospital
Department Name
Neonatology
Contact Person Name
Mirjam van Weissenbruch
Contact Person Email
m.vanweissenbruch@vumc.nl
Site Name
Meander Medisch Centrum
Department Name
Neonatology
Contact Person Name
Clemens Meijssen
Contact Person Email
cb.meijssen@meandermc.nl
Site Name
Erasmus Universitair Medisch Centrum Rotterdam (Erasmus MC)
Department Name
Neonatology
Contact Person Name
Gerbrich van den Bosch
Contact Person Email
g.vandenbosch@erasmusmc.n
Site Name
OLVG
Department Name
Neonatology
Contact Person Name
Sophie van der Schoor
Contact Person Email
s.r.d.vanderschoor@olvg.nl
Site Name
Albert Schweitzer Ziekenhuis
Department Name
Neontatology
Contact Person Name
Miranda de Jong
Contact Person Email
m.dejong@asz.nl

Austria

Earliest CTIS Part Ii Submission Date
22-08-2024
Latest Decision Or Authorization Date
14-01-2025
Processing Time Days
145
Number Of Sites
3
Number Of Participants
49

Sites

Site Name
Universitätsklinik für Kinder- und Jugendheilkunde
Department Name
Klinische Abteilung für Neonatologie
Contact Person Name
Gerhard Pichler
Contact Person Email
gerhard.pichler@medunigraz.at
Site Name
Medizinische Universität Wien
Department Name
Klinische Abteilung für Neonatologie, Pädiatrische Intensivmedizin und Neuropädiatrie
Contact Person Name
Katrin Klebermass-Schehof
Site Name
Universitätsklinik für Kinder- und Jugendheilkunde der PMU
Department Name
Division für Neonatologie
Contact Person Name
Martin Wald
Contact Person Email
neooffice@salk.at

Estonia

Earliest CTIS Part Ii Submission Date
22-08-2024
Latest Decision Or Authorization Date
16-09-2024
Processing Time Days
25
Number Of Sites
2
Number Of Participants
14

Sites

Site Name
Tartu University Hospital
Department Name
Neonatology
Contact Person Name
Tuuli Metsvaht
Contact Person Email
tuuli.metsvaht@kliinikum.ee
Site Name
East Tallinn Central Hospital
Department Name
Neonatology
Contact Person Name
Pille Andresson
Contact Person Email
pille.andresson@itk.ee

Belgium

Earliest CTIS Part Ii Submission Date
22-08-2024
Latest Decision Or Authorization Date
06-08-2025
Processing Time Days
349
Number Of Sites
2
Number Of Participants
29

Sites

Site Name
CHR de la Citadelle
Department Name
Neonatology
Contact Person Name
Renaud Viellevoye
Site Name
KU Leuven
Department Name
Neonatology
Contact Person Name
Gunnar Naulaers
Contact Person Email
gunnar.naulaers@uzleuven.be

Sponsor

Primary sponsor

Full Name
Universitaetsklinikum Tuebingen AöR
Organisation Type
Hospital/Clinic/Other health care facility
Country Of Registered Address
Germany

Investigational products

Investigational Product Name
ACEPURIN, poeder voor infusievloeistof 1g/100 ml
Active Substance
Allopurinol sodium
Modality
Small molecule
Routes Of Administration
INTRAVENOUS USE
Route
Intravenous
Authorisation Status
Authorised (marketing authorisation RVG 09974 in NL)
Orphan Designation
Yes
Maximum Dose
30 mg/kg
Investigational Product Name
MANNITOL
Active Substance
Mannitol
Modality
Small molecule
Routes Of Administration
SOLUTION FOR INFUSION
Route
Infusion
Authorisation Status
Authorised
Maximum Dose
30 mg/kg

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