Clinical trial • Phase III • Psychiatry

trospium chloride; xanomeline tartrate for Agitation associated with Alzheimer's disease

Phase III trial of trospium chloride; xanomeline tartrate for Agitation associated with Alzheimer's disease.

Overview

Trial Therapeutic Area
Psychiatry
Trial Disease
Agitation associated with Alzheimer's disease
Trial Stage
Phase III
Drug Modality
Small molecule

Key dates

Initial CTIS Submission Date
30-06-2025
First CTIS Authorization Date
20-10-2025

Trial design

Randomised, placebo (karxt matching placebo and karx-ec matching placebo); dose and schedule not specified in available documents.-controlled Phase III trial across 51 sites in Romania, Bulgaria, Portugal and others.

Randomised
Yes
Comparator
Placebo (KarXT matching Placebo and KarX-EC matching Placebo); dose and schedule not specified in available documents.
Target Sample Size
251

Eligibility

Recruits 251 Participants are individuals with Alzheimer’s disease (cognitive impairment) identified as a vulnerable population. A caregiver/study partner must be identified; the caregiver is required to attend visits, oversee compliance and provide informed consent (IC) for participation. The trial includes subject information sheets, informed consent forms, study-partner ICFs and assent documents (e.g., Adult Assent) and these materials are available in multiple country/language versions (examples in the document list include EN, BG, PT, GR, HR, RO, ES)..

Vulnerable Population
Participants are individuals with Alzheimer’s disease (cognitive impairment) identified as a vulnerable population. A caregiver/study partner must be identified; the caregiver is required to attend visits, oversee compliance and provide informed consent (IC) for participation. The trial includes subject information sheets, informed consent forms, study-partner ICFs and assent documents (e.g., Adult Assent) and these materials are available in multiple country/language versions (examples in the document list include EN, BG, PT, GR, HR, RO, ES).

Inclusion criteria

  • {"criterion_text":"- A diagnosis of Alzheimer’s disease (AD) in accordance with the 2024 Alzheimer’s Association criteria with one of the the following confirmations of AD pathology: \t- Historical evidence of AD diagnosis with amyloid positron emission tomography (PET), Aβ42/40 ratio in CSF, pTau181/Aβ42 ratio in CSF or pTau217/Aβ42 ratio in plasma using an Health Authority (HA)-authorized diagnostic assay. \t- If no historical evidence available: A. A plasma biomarker will be assessed for eligibility if allowed per regulatory requirements. The test cutoff(s) will be based on diagnostic use approval. B. If a plasma biomarker assay cannot be used or if the assay result is inconclusive, conduct one the following: o Amyloid PET o Aβ42/40 ratio or pTau181/Aβ42 ratio in CSF using an HA-authorized diagnostic assay\n- Mini-Mental State Examination (MMSE) score of 5 to 22, inclusive, at Screening (Visit 1)\n- Have one identified caregiver who should have sufficient contact (approximately 10 hours a week or more) and is willing to:  Attend all visits and report on participant’s status Oversee participant compliance with medication and study procedures  Participate in the study assessments and provide IC to participate in the study\n- History of agitation that meets the International Psychogeriatric Association (IPA) consensus definition for agitation in cognitive disorders with onset at least two weeks prior to Screening (Visit 1).\n- AD participants are required to have NPI/NPI-NH Agitation/Aggression score ≥ 4 at Screening (Visit 1) and Baseline (Visit 2).\n- CGI-S ≥ 4, as related to agitation, at Screening (Visit 1) and Baseline (Visit 2)\n- At least 1 of the following 3 criteria must be established from the CMAI-IPA at Screening (Visit 1) and Baseline (Visit 2; CMAI-IPA Physical/Verbal Aggression Positivity):  1 or more aggressive behaviors occurring several times per week  2 or more aggressive behaviors occurring once or twice per week  3 or more aggressive behaviors occurring less than once per week"}

Exclusion criteria

  • {"criterion_text":"- Medical Conditions  Agitation symptoms that are primarily attributable to a condition other than the AD causing the dementia  History of bipolar disorder, schizophrenia, or schizoaffective disorder  History of (or at high risk for) urinary retention, gastric retention, or narrow-angle glaucoma as evaluated by the Investigator  Risk of suicidal behavior during the study as determined by the Investigator’s clinical assessment and/or C-SSR\n- Prior/Concomitant Therapy - Recent history of receiving monoamine oxidase inhibitors, anticonvulsants (eg, lamotrigine, divalproex), mood stabilizers (eg, lithium), tricyclic antidepressants (eg, imipramine, desipramine), or any other psychoactive medications except for as needed anxiolytics (eg, lorazepam)  Selective serotonin reuptake inhibitors and serotonin norepinephrine reuptake inhibitors taken at a stable dose for at least 8 weeks prior to Screening (Visit 1) may be permitted  Mirtazapine or trazodone may be used as a hypnotic if started at least 8 weeks prior to Screening (Visit 1)\n- Other protocol-defined Inclusion/Exclusion criteria apply."}

Endpoints

Primary endpoints

  • {"endpoint_text":"- Change from baseline to the end of treatment on the CMAI-IPA total score compared with placebo.","definition_or_measurement_approach":"Change from baseline to end of treatment measured by the Cohen-Mansfield Agitation Inventory – International Psychogeriatric Association (CMAI-IPA) total score; comparison versus placebo."}

Secondary endpoints

  • {"endpoint_text":"- Change from baseline to the end of treatment on the CGI-S as it relates specifically to agitation compared with placebo.","definition_or_measurement_approach":"Change from baseline to end of treatment measured by the Clinical Global Impressions – Severity (CGI-S) score specifically related to agitation; comparison versus placebo."}

Recruitment

Planned Sample Size
251
Recruitment Window Months
37
Consent Approach
Informed consent is obtained via subject information sheets and informed consent forms. For this vulnerable population (participants with AD), a caregiver/study partner is required and is expected to provide informed consent; study-partner ICFs and adult assent forms are included. Consent/assent documentation exists in multiple language/country-specific versions (examples in the document list: EN, BG, PT, GR, HR, RO, ES).

Methods

  • Site-based recruitment using study-site recruitment materials: PI-to-patient/participant letters, recruitment posters, study intro trifolds and caregiver fact sheets. Country-specific recruitment materials/documents are provided (document list includes K1/K2 recruitment materials for BG, PT, GR, ES, HR, RO).

Geography

Total Number Of Sites
51
Total Number Of Participants
103

Romania

Earliest CTIS Part Ii Submission Date
11-07-2025
Latest Decision Or Authorization Date
21-04-2026
Processing Time Days
284
Number Of Sites
13
Number Of Participants
25

Sites

Site Name
Spitalul Clinic De Psihiatrie Prof.Dr.Alexandru Obregia
Department Name
Psychiatry
Contact Person Name
Laura Cristina Dolis
Contact Person Email
drcristinadolis@gmail.com
Site Name
Institutul De Psihiatrie Socola Iasi
Department Name
Psychiatry
Contact Person Name
Cristinel Stefanescu
Contact Person Email
cristinel.stefanescu@gmail.com
Site Name
Centrul de Evaluare și Tratament a Toxicodependenței pentru Tineri Sf.Stelian
Department Name
Psychiatry
Contact Person Name
Tr Barbu
Contact Person Email
trabar98@yahoo.com
Site Name
Spitalul Clinic De Psihiatrie Si Neurologie Brasov
Department Name
Psychiatry
Contact Person Name
Petru Ifteni
Contact Person Email
relatiicupublicul@spnbrasov.ro
Site Name
Spitalul Clinic De Psihiatrie Dr. Gheorghe Preda Sibiu
Department Name
Psychiatry
Contact Person Name
Ciprian Bacila
Contact Person Email
bacila_c@yahoo.com
Site Name
Spitalul Clinic De Psihiatrie Prof.Dr.Alexandru Obregia
Department Name
Psychiatry
Contact Person Name
Corina Mihaela Nicolae
Contact Person Email
corina_panzaru@yahoo.com
Site Name
Spitalul Clinic De Psihiatrie Prof.Dr.Alexandru Obregia
Department Name
Psychiatry
Contact Person Name
Mihnea Manea
Contact Person Email
maneamihnea@gmail.com
Site Name
Spitalul Clinic De Psihiatrie Prof.Dr.Alexandru Obregia
Department Name
Psychiatry
Contact Person Name
Valentin Matei
Contact Person Email
valipmatei@yahoo.com
Site Name
Spitalul Clinic De Psihiatrie Prof.Dr.Alexandru Obregia
Department Name
Psychiatry
Contact Person Name
Simona Trifu
Contact Person Email
simonatrifu@yahoo.com
Site Name
Spitalul Clinic De Psihiatrie Prof.Dr.Alexandru Obregia
Department Name
Psychiatry
Contact Person Name
Adela Ciobanu
Contact Person Email
adela.ciobanu@yahoo.com
Site Name
Spitalul Universitar De Urgenta Militar Central Dr. Carol Davila
Department Name
Psychiatry
Contact Person Name
Octavian Vasiliu
Contact Person Email
octavvasiliu@yahoo.com
Site Name
Spitalul Clinic De Psihiatrie Prof.Dr.Alexandru Obregia
Department Name
Psychiatry
Contact Person Name
Mihaela Cleopatra Rosca
Contact Person Email
mihaelarosca@gmail.com
Site Name
Cai Ferate Clinical Hospital Constanta
Department Name
Neurology
Contact Person Name
Ana Maria Ionescu
Contact Person Email
iuliusana@gmail.com

Bulgaria

Earliest CTIS Part Ii Submission Date
10-10-2025
Latest Decision Or Authorization Date
20-04-2026
Processing Time Days
192
Number Of Sites
5
Number Of Participants
10

Sites

Site Name
Medical Center Saint Naum EOOD
Department Name
Psychiatry
Contact Person Name
Asen Karadaliev
Contact Person Email
xxxx@xxxx.com
Site Name
Outpatient Clinic for Indiv. Practice for Spec.Med. Care in Psychiatry-Dr.Madlena Dimitrova Borisova
Department Name
Psychiatry
Contact Person Name
Madlena Borisova
Site Name
Medical Center Medconsult Pleven OOD
Department Name
Psychiatry
Contact Person Name
Maria Aleksandrova
Contact Person Email
xxxx@xxxx.com
Site Name
Mental Health Center Sofia EOOD
Department Name
Department for active treatment of individuals with severe psychiatric disorders – Psychiatry, Level
Contact Person Name
Emil Grashnov
Contact Person Email
xxxx@xxxx.com
Site Name
Diagnostics-Consultancy Center Mladost M Varna OOD
Department Name
Psychiatry
Contact Person Name
Hristo Kozhuharov
Contact Person Email
mcoffice@mkmladost.com

Portugal

Earliest CTIS Part Ii Submission Date
06-10-2025
Latest Decision Or Authorization Date
17-04-2026
Processing Time Days
193
Number Of Sites
6
Number Of Participants
8

Sites

Site Name
CNS Saude Lda.
Department Name
Neurology
Contact Person Name
Camila Nobrega
Contact Person Email
xxxxx@xxxx.com
Site Name
Unidade Local De Saude De Matosinhos E.P.E.
Department Name
Neurology
Contact Person Name
Vítor Cruz
Contact Person Email
investigacao@ulsm.min-saude.pt
Site Name
Unidade Local De Saude De Santa Maria E.P.E.
Department Name
Neurology
Contact Person Name
Ana Verdelho
Contact Person Email
xxxxx@xxxx.com
Site Name
Unidade Local De Saude Do Alto Ave E.P.E.
Department Name
Neurology
Contact Person Name
Joana Meireles
Site Name
Unidade Local De Saude De Coimbra E.P.E.
Department Name
Neurology
Contact Person Name
Maria Isabel Santana
Contact Person Email
xxxxx@xxxx.com
Site Name
Unidade Local De Saude De Coimbra E.P.E.
Department Name
Neurology
Contact Person Name
Maria Isabel Santana
Contact Person Email
xxxxx@xxxx.com

Croatia

Earliest CTIS Part Ii Submission Date
22-09-2025
Latest Decision Or Authorization Date
21-04-2026
Processing Time Days
211
Number Of Sites
4
Number Of Participants
13

Sites

Site Name
KBC Split
Department Name
Psychiatry
Contact Person Name
Trpimir Glavina
Contact Person Email
psihijatrija@kbsplit.hr
Site Name
Clinical Hospital Centre Rijeka
Department Name
Psychiatry
Contact Person Name
Vladimir Sabljić
Contact Person Email
vladimir.sabljic@ri.t-com.hr
Site Name
KBC Zagreb
Department Name
Neurology
Contact Person Name
Nataša Klepac
Contact Person Email
natasaklepac@gmail.com
Site Name
Opca Bolnica Varazdin
Department Name
Neurology
Contact Person Name
Spomenka Kiđemet Piskač
Contact Person Email
spiskac@gmail.com

Greece

Earliest CTIS Part Ii Submission Date
11-07-2025
Latest Decision Or Authorization Date
17-04-2026
Processing Time Days
280
Number Of Sites
10
Number Of Participants
18

Sites

Site Name
Eginitio Hospital
Department Name
A’ Department of Neurology
Contact Person Name
Nikolaos Scarmeas
Contact Person Email
ns257@columbia.edu
Site Name
General University Hospital Of Patras
Department Name
Department of Neurology
Contact Person Name
John Ellul
Contact Person Email
ellul@upatras.gr
Site Name
Eginitio Hospital
Department Name
First Department of Psychiatry
Contact Person Name
Nikolaos Stefanis
Contact Person Email
nistefan@med.uoa.gr
Site Name
University General Hospital Of Ioannina
Department Name
Department of Neurology
Contact Person Name
Spyridon Konitsiotis
Contact Person Email
skonitso@uoi.gr
Site Name
University General Hospital Attikon
Department Name
2nd Department of Neurology
Contact Person Name
Georgios Tsivgoulis
Contact Person Email
tsivgoulisgiorg@yahoo.gr
Site Name
Euromedica General Clinic Of Thessaloniki
Department Name
Neurological Department
Contact Person Name
Magdalini Tsolaki
Contact Person Email
tsolakim@gmail.com
Site Name
Henry Dunant Hospital Center
Department Name
2nd Neurological Clinic
Contact Person Name
Konstantina Yiannopoulou
Contact Person Email
k.giannopoulou.14@hotmail.com
Site Name
Athens Medical Center S.A.
Department Name
Memory Clinic
Contact Person Name
Ioannis Papatriantafyllou
Contact Person Email
ipapatriantafyllou@gmail.com
Site Name
Eginitio Hospital
Department Name
A’ Department of Neurology
Contact Person Name
Nikolaos Scarmeas
Contact Person Email
ns257@columbia.edu
Site Name
General University Hospital Of Patras
Department Name
Department of Neurology
Contact Person Name
John Ellul
Contact Person Email
ellul@upatras.gr

Spain

Earliest CTIS Part Ii Submission Date
14-08-2025
Latest Decision Or Authorization Date
21-04-2026
Processing Time Days
281
Number Of Sites
13
Number Of Participants
29

Sites

Site Name
Hospital Universitario Rio Hortega
Department Name
Neurología
Contact Person Name
Juan Muñoz Sanchez
Contact Person Email
jlmusa@icloud.com
Site Name
Hospital Universitario Virgen De La Victoria
Department Name
Neurología
Contact Person Name
Carlos De La Cruz Cosme
Contact Person Email
XXXX@XXXX.XX
Site Name
Oroitu S.L.
Department Name
Neurología
Contact Person Name
MANUEL FERNANDEZ
Contact Person Email
mfernandezm@oroitu.com
Site Name
Consorci Sanitari De Terrassa
Department Name
Neurología
Contact Person Name
Jerzy Krupinski
Contact Person Email
jkrupinski@mutuaterrassa.es
Site Name
Hospital Clinico San Carlos
Department Name
Neurología
Contact Person Name
Jordi Matias Guiu
Site Name
Hospital General Universitario De Elche
Department Name
gonzalez_glocab@gva.es
Contact Person Name
Maria Gloria González Caballero
Contact Person Email
gonzalez_glocab@gva.es
Site Name
Hospital Ruber Juan Bravo
Department Name
Neurología
Contact Person Name
Juan Lopez Lozano
Contact Person Email
XXXX@XXXX.XX
Site Name
Hospital Victoria Eugenia De La Cruz Roja Espanola
Department Name
Neurología
Contact Person Name
Felix Viñuela Fernandez
Contact Person Email
XXXX@XXXX.XX
Site Name
Hospital Universitario De Salamanca
Department Name
Neurología
Contact Person Name
Angel Luis Montejo
Contact Person Email
amontejo@usal.es
Site Name
Clinica Universidad De Navarra
Department Name
Neurología
Contact Person Name
Mario Riverol Fernandez
Contact Person Email
mriverol@unav.es
Site Name
Clinica Montecanal S.L.
Department Name
Neurología
Contact Person Name
Antonio Oliveros-Cid
Contact Person Email
XXXX@XXXX.XX
Site Name
Hospital General Universitario De Elche
Department Name
Neurología
Contact Person Name
Maria Gloria González Caballero
Contact Person Email
gonzalez_glocab@gva.es
Site Name
Hospital Universitario Rio Hortega
Department Name
Neurología
Contact Person Name
Juan Muñoz Sanchez
Contact Person Email
jlmusa@icloud.com

Sponsor

Primary sponsor

Full Name
Bristol-Myers Squibb Services Unlimited Company
Organisation Type
Pharmaceutical company
Country Of Registered Address
Ireland

Contract research organisations

Name
Syneos Health Inc.
Responsibilities
Subject Eligibility Review
Name
Iqvia Holdings Inc.
Responsibilities
Site Payments

Third parties

  • {"country":"United States","full_name":"Syneos Health Inc.","duties_or_roles":"Subject Eligibility Review","organisation_type":"Pharmaceutical company"}
  • {"country":"Switzerland","full_name":"Labcorp Central Laboratory Services SARL","duties_or_roles":"Safety Laboratory testing and pTau217/AB42, pTau181/AB42, AB42/40 Biomarker testing","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Iqvia Holdings Inc.","duties_or_roles":"Site Payments","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Greenphire LLC","duties_or_roles":"Provides electronic payments, travel arrangements,electronic study-related comunications to patients","organisation_type":"Non-Pharmaceutical company"}
  • {"country":"India","full_name":"Accenture Solutions Private Limited","duties_or_roles":"Pharmacovigilance duties: Medical review and Cases Data Entry","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Medidata Solutions Inc.","duties_or_roles":"Data Management Platform","organisation_type":"Non-Pharmaceutical company"}
  • {"country":"United States","full_name":"Signant Health LLC","duties_or_roles":"PRO/COA management, rater training, and supply of electronic devices for the collection of eCOA assessments","organisation_type":"Pharmaceutical company"}

Investigational products

Investigational Product Name
KarXT
Active Substance
trospium chloride; xanomeline tartrate
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Authorisation Status
Authorised
Investigational Product Name
KarX-EC
Active Substance
xanomeline tartrate
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Authorisation Status
Authorised
Investigational Product Name
KarXT matching Placebo
Modality
Other
Authorisation Status
Not applicable
Investigational Product Name
KarX-EC matching Placebo
Modality
Other
Authorisation Status
Not applicable
Combination Treatment
Yes

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