Clinical trial • Phase II • Oncology

INAVOLISIB for Solid tumor

Phase II trial of INAVOLISIB for Solid tumor. 499 participants.

Overview

Trial Therapeutic Area
Oncology
Trial Disease
Solid tumor
Trial Stage
Phase II
Drug Modality
Small molecule|Monoclonal antibody
Paediatric Trial
Yes

Key dates

Initial CTIS Submission Date
10-06-2024
First CTIS Authorization Date
12-07-2024

Trial design

Phase II trial in Italy, Germany, Portugal and others.

Biomarker Stratified
True, Somatic tumor genomic alterations (alteration/biomarker-positive cohorts; e.g. RET, NTRK, ALK, PIK3CA, KRAS G12C, BRAF, ROS1 as indicated by cohort-specific documents)
Target Sample Size
499

Eligibility

Recruits 499 paediatric patients.

Pregnancy Exclusion
Pregnant or breastfeeding, or intending to become pregnant during the study
Vulnerable Population
Vulnerable populations are included (pediatric participants). Age-specific performance criteria and multiple paediatric age cohorts are specified (participants aged <16 years, 16 to <18 years, etc.). Assent and parental consent procedures are provided: multiple assent and parent/guardian ICF documents are listed for cohorts (e.g. Assent 3-11 yr, 7-11 yr, 12-17 yr and corresponding parent ICFs), indicating minors require parental consent and age-appropriate assent forms.

Inclusion criteria

  • {"criterion_text":"- Histologically or cytologically confirmed diagnosis of advanced and unresectable or metastatic solid malignancy"}
  • {"criterion_text":"- Measurable disease as defined by Response Evaluation Criteria in Solid Tumors, Version 1.1 (RECIST v1.1), Response Assessment in Neuro-Oncology (RANO) criteria, or International Neuroblastoma Response Criteria (INRC)"}
  • {"criterion_text":"- Performance status as follows: Participants aged ≥ 18 years: Eastern Cooperative Oncology Group (ECOG) Performance Status 0-2; Participants aged 16 to < 18 years: Karnofsky score ≥ 50%; Participants aged < 16 years: Lansky score ≥ 50%"}
  • {"criterion_text":"- For participants aged ≥ 18 and <18 years: adequate hematologic and end-organ function"}
  • {"criterion_text":"- Disease progression on prior treatment, or previously untreated disease with no available acceptable treatment"}
  • {"criterion_text":"- Adequate recovery from most recent systemic or local treatment for cancer"}

Exclusion criteria

  • {"criterion_text":"- Current participation or enrollment in another therapeutic clinical trial"}
  • {"criterion_text":"- Any anticancer treatment within 2 weeks prior to start of study treatment (Please refer to the cohort-specific eligibility criteria for requirements on enrollment, if applicable)"}
  • {"criterion_text":"- Whole brain radiotherapy within 14 days prior to start of study treatment"}
  • {"criterion_text":"- Stereotactic radiosurgery within 7 days prior to start of study treatment"}
  • {"criterion_text":"- Pregnant or breastfeeding, or intending to become pregnant during the study"}
  • {"criterion_text":"- History of or concurrent serious medical condition or abnormality in clinical laboratory tests that, in the investigator's judgment, precludes the participant's safe participation in and completion of the study or confounds the ability to interpret data from the study"}

Endpoints

Primary endpoints

  • {"endpoint_text":"- 1 Independent Review Committee (IRC)-assessed objective response rate (ORR) based on confirmed (≥4 weeks after initial documentation of response) objective response (per RECIST v1.1)","definition_or_measurement_approach":"IRC-assessed ORR based on confirmed objective response (confirmation ≥4 weeks after initial documentation of response), evaluated per RECIST v1.1"}

Secondary endpoints

  • {"endpoint_text":"- 1 IRC-assessed duration of response (DOR), clinical benefit rate (CBR), and progression-free survival (PFS) per RECIST v1.1","definition_or_measurement_approach":"Evaluated by IRC per RECIST v1.1"}
  • {"endpoint_text":"- 2 Investigator (INV)-assessed ORR, DOR, CBR, and PFS per RECIST v1.1","definition_or_measurement_approach":"Assessed by investigator per RECIST v1.1"}
  • {"endpoint_text":"- 3 IRC- and INV-assessed time to CNS progression per RECIST v1.1","definition_or_measurement_approach":"Time to CNS progression measured per RECIST v1.1 by IRC and investigator"}
  • {"endpoint_text":"- 4 Overall survival (OS)","definition_or_measurement_approach":"Overall survival measured as time from baseline to death from any cause"}
  • {"endpoint_text":"- 5 Cohorts A, B, C, D, I, J, and K: IRC-assessed CNS-ORR, CNS-DOR, CNS-CBR, and CNS-PFS per RANO","definition_or_measurement_approach":"IRC assessment per RANO criteria for CNS endpoints"}
  • {"endpoint_text":"- 6 Cohorts A, B, C, D, I, J, and K: INV-assessed CNS-ORR, CNS-DOR, CNS-CBR, and CNS-PFS per RANO","definition_or_measurement_approach":"Investigator assessment per RANO criteria for CNS endpoints"}
  • {"endpoint_text":"- 7 Cohorts A, B, C, D, E, H, I, J, K, L, M, and N: IRC-assessed ORR, DOR, CBR, and PFS per International Neuroblastoma Response Criteria (INRC)","definition_or_measurement_approach":"IRC assessment per INRC for neuroblastoma cohorts"}
  • {"endpoint_text":"- 8 Cohorts A, B, C, D, E, H, I, J, K, L, M, and N: INV-assessed ORR, DOR, CBR, and PFS per INRC","definition_or_measurement_approach":"Investigator assessment per INRC for neuroblastoma cohorts"}
  • {"endpoint_text":"- 9 Cohorts A, B, C, D, I, J, and K: IRC-assessed IC-ORR, IC-DOR, IC-CBR, IC-PFS rate per RECIST v1.1","definition_or_measurement_approach":"IRC assessment of intracranial (IC) endpoints per RECIST v1.1"}
  • {"endpoint_text":"- 10. Cohorts A, B, C, D, I, J, and K: INV-assessed IC-ORR, IC-DOR, IC-CBR, IC-PFS per RECIST v1.1","definition_or_measurement_approach":"Investigator assessment of intracranial endpoints per RECIST v1.1"}
  • {"endpoint_text":"- 11. Descriptive endpoint of time to confirmed deterioration, change from baseline, proportion of patients with a clinical meaningful change on the Global Health Status, Physical Functioning, and Role Functioning scores from the European Organisation for Research and Treatment of Cancer (EORTC) QLQ-C30","definition_or_measurement_approach":"Patient-reported outcomes measured using EORTC QLQ-C30 (Global Health Status, Physical Functioning, Role Functioning); time to confirmed deterioration and proportion with clinically meaningful change"}
  • {"endpoint_text":"- 12. Descriptive endpoint of time to confirmed symptom onset or worsening from tumor-related symptom scores from the EORTC QLQ-C30 and EORTC IL71","definition_or_measurement_approach":"Symptom scores from EORTC QLQ-C30 and EORTC IL71; time to confirmed symptom onset or worsening"}
  • {"endpoint_text":"- 13. Incidence, type, and severity of adverse events (based on the NCI CTCAE v5.0), including serious adverse events","definition_or_measurement_approach":"Adverse events graded per NCI CTCAE v5.0; incidence, type and severity summarized"}
  • {"endpoint_text":"- 14. Cohort K: for pediatric patients - evaluate the acceptability and palatability of pralsetinib with Acceptability Survey scores on Day 1 of Cycle 1","definition_or_measurement_approach":"Acceptability Survey scores on Day 1 of Cycle 1 for pralsetinib in pediatric cohort K"}

Recruitment

Digital Remote Recruitment
True, remote NGS prescreening documents are listed (e.g. "L1_SIS and ICF 7-11 yr NGS remote prescreening", "L1_SIS and ICF 12-17 yr NGS remote prescreening"), indicating remote/digital prescreening methods
Planned Sample Size
499
Recruitment Window Months
137
Consent Approach
Age-appropriate informed consent and assent processes are provided. Parental/guardian informed consent is required for minors; assent forms are provided for paediatric age groups (documents listed for 3-11 yr, 7-11 yr, 12-17 yr cohorts and corresponding parent ICFs). Separate ICFs and parent documents for paediatric and adult cohorts and remote prescreening ICFs are included.

Geography

Total Number Of Sites
37
Total Number Of Participants
407

Italy

Earliest CTIS Part Ii Submission Date
26-06-2024
Latest Decision Or Authorization Date
30-10-2025
Processing Time Days
491
Number Of Sites
7
Number Of Participants
100

Sites

Site Name
Fondazione IRCCS Istituto Nazionale Dei Tumori
Department Name
S.C. MEDICINA ONCOLOGICA 1
Contact Person Name
Silvia Damian
Site Name
Fondazione Policlinico Universitario Agostino Gemelli IRCCS
Department Name
UOS Fase I
Contact Person Name
Gennaro Daniele
Site Name
Azienda Ospedaliera Universitaria Citta Della Salute E Della Scienza Di Torino
Department Name
Osp. Infantile Regina Margherita
Contact Person Name
Franca Fagioli
Contact Person Email
franca.fagioli@unito.it
Site Name
Bambino Gesu Childrens Hospital
Department Name
Dipartimento di Onco-Ematologia Pediatrica
Contact Person Name
Franco Locatelli
Contact Person Email
franco.locatelli@opbg.net
Site Name
Azienda Socio Sanitaria Territoriale Degli Spedali Civili Di Brescia
Department Name
U.O. Oncologia Medica
Contact Person Name
Salvatore Grisanti
Contact Person Email
grisanti.salvatore@gmail.com
Site Name
Azienda Ospedaliera Universitaria Senese
Department Name
U.O.C. Immunoterapia Oncologica
Contact Person Name
Michele Maio
Contact Person Email
mmaiocro@gmail.com
Site Name
Fondazione IRCCS Istituto Nazionale Dei Tumori
Department Name
S.C. Oncologia Pediatrica
Contact Person Name
Michela Casanova

Germany

Earliest CTIS Part Ii Submission Date
26-06-2024
Latest Decision Or Authorization Date
30-10-2025
Processing Time Days
491
Number Of Sites
2
Number Of Participants
7

Sites

Site Name
SLK-Kliniken Heilbronn GmbH
Department Name
Klinik für Innere Medizin III
Contact Person Name
Uwe Martens
Contact Person Email
medklinik3@slk-kliniken.de
Site Name
Universitaetsklinikum Essen AöR
Department Name
Westdeutsches Tumorzentrum
Contact Person Name
Martin Schuler
Contact Person Email
Martin.Schuler@uk-essen.de

Portugal

Earliest CTIS Part Ii Submission Date
26-06-2024
Latest Decision Or Authorization Date
29-10-2025
Processing Time Days
490
Number Of Sites
1
Number Of Participants
13

Sites

Site Name
Instituto Portugues De Oncologia Do Porto Francisco Gentil E.P.E.
Department Name
Serviço de Oncologia Médica
Contact Person Name
Júlio Oliveira

Belgium

Earliest CTIS Part Ii Submission Date
26-06-2024
Latest Decision Or Authorization Date
30-10-2025
Processing Time Days
491
Number Of Sites
5
Number Of Participants
50

Sites

Site Name
UZ GENT
Department Name
Pediatric Hematology - Oncology
Contact Person Name
Bram De Wilde
Contact Person Email
Bram.DeWilde@uzgent.be
Site Name
Cliniques Universitaires Saint-Luc
Department Name
Medical oncology
Contact Person Name
Cedric Van Marcke
Site Name
Grand Hôpital de Charleroi - Site Les Viviers
Department Name
Oncology & Hematology
Contact Person Name
Jean-Luc Canon
Contact Person Email
jean-luc.canon@ghdc.be
Site Name
Antwerp University Hospital
Department Name
Multidisciplinary Oncology Centre
Contact Person Name
Hans Prenen
Contact Person Email
hans.prenen@uza.be
Site Name
UZ Leuven
Department Name
Oncology
Contact Person Name
Sabine Tejpar
Contact Person Email
sabine.tejpar@uzleuven.be

Denmark

Earliest CTIS Part Ii Submission Date
26-06-2024
Latest Decision Or Authorization Date
28-10-2025
Processing Time Days
489
Number Of Sites
1
Number Of Participants
8

Sites

Site Name
Rigshospitalet
Department Name
Onkologisk Klinik
Contact Person Name
Kristoffer Rohrberg

Poland

Earliest CTIS Part Ii Submission Date
26-06-2024
Latest Decision Or Authorization Date
09-12-2025
Processing Time Days
531
Number Of Sites
4
Number Of Participants
60

Sites

Site Name
Narodowy Instytut Onkologii Im. Marii Sklodowskiej-Curie Panstwowy Instytut Badawczy
Department Name
Klinika Nowotworów Płuca i Klatki Piersiowej, Klinika Gin Onkologicznej, Oddział Badań Wczesnych Faz
Contact Person Name
Maciej Krzakowski
Site Name
Uniwersyteckie Centrum Kliniczne (Gdansk)
Department Name
Klinika Onkoligii i Radioterapii
Contact Person Name
Rafał Dziadziuszko
Contact Person Email
onkol@gumed.edu.pl
Site Name
Uniwersyteckie Centrum Kliniczne (Gdansk) - pediatrics
Department Name
Klinika Pediatrii, Hematologii i Onkologii
Contact Person Name
Rafał Dziadziuszko
Contact Person Email
onkol@gumed.edu.pl
Site Name
Narodowy Instytut Onkologii Im. Marii Sklodowskiej-Curie Panstwowy Instytut Badawczy (Warsaw)
Department Name
Klinika Onkologii i Radioterapii
Contact Person Name
Maciej Krzakowski

Spain

Earliest CTIS Part Ii Submission Date
26-06-2024
Latest Decision Or Authorization Date
31-10-2025
Processing Time Days
492
Number Of Sites
11
Number Of Participants
95

Sites

Site Name
Hospital Infantil Universitario Nino Jesus
Department Name
Oncología
Contact Person Name
Alba Rubio San Simón
Contact Person Email
Alba.rubio@salud.madrid.org
Site Name
Hospital Universitario Hm Sanchinarro
Department Name
Oncología
Contact Person Name
Irene Moreno Candilejo
Contact Person Email
irene.moreno@startmadrid.com
Site Name
Hospital Universitario Y Politecnico La Fe
Department Name
Oncología
Contact Person Name
Javier Caballero Daroqui
Contact Person Email
daroqui@gmail.com
Site Name
Clinica Universidad De Navarra (Pamplona)
Department Name
Oncología
Contact Person Name
María Luisa Sánchez Lorenzo
Contact Person Email
lsanchezl@unav.es
Site Name
Hospital Universitario Fundacion Jimenez Diaz
Department Name
Oncología
Contact Person Name
Victor Moreno García
Contact Person Email
victor.moreno@startmadrid.com
Site Name
Hospital Universitari Vall D Hebron
Department Name
Oncología
Contact Person Name
Lucas Moreno Martín
Contact Person Email
lucas.moreno@vallhebron.cat
Site Name
Clinica Universidad De Navarra (Madrid)
Department Name
Oncología
Contact Person Name
María Luisa Sánchez Lorenzo
Contact Person Email
lsanchezl@unav.es
Site Name
Sant Joan De Deu Barcelona Hospital
Department Name
Oncología
Contact Person Name
Jaume Mora Graupera
Contact Person Email
jaume.mora@sjd.es
Site Name
Fir Huvh Fundacio Institut De Recerca Hospital Universitari Vall De Hebron
Department Name
Oncología
Contact Person Name
Elena Garralda Cábanas
Contact Person Email
egarralda@vhio.net
Site Name
Hospital Universitario La Paz
Department Name
Oncología
Contact Person Name
Javier De Castro Carpeno
Site Name
Hospital Universitario 12 De Octubre
Department Name
Oncología
Contact Person Name
Luis Paz- Arez Rodriguez
Contact Person Email
lpazaresr@seom.org

France

Earliest CTIS Part Ii Submission Date
26-06-2024
Latest Decision Or Authorization Date
02-02-2026
Processing Time Days
586
Number Of Sites
6
Number Of Participants
74

Sites

Site Name
Institut Bergonie
Department Name
Medical Oncology
Contact Person Name
Veronique DEBIEN
Contact Person Email
v.debien@bordeaux.unicancer.fr
Site Name
Centre Oscar Lambret
Department Name
Oncology
Contact Person Name
Sandra RAIMBAULT
Contact Person Email
s-raimbault@o-lambret.fr
Site Name
Institut Gustave Roussy
Department Name
Drug Development Department (DITEP) – U981 INSERM
Contact Person Name
Christophe MASSARD
Site Name
Centre Hospitalier Regional De Marseille
Department Name
Pediatric Immunology, Hematology and Oncology Department
Contact Person Name
Nicolas Andre
Contact Person Email
nicolas.andre@ap-hm.fr
Site Name
Institut Universitaire Du Cancer Toulouse-Oncopole
Department Name
Medical Oncology
Contact Person Name
Carlos Alberto Gomez Roca
Site Name
Centre Leon Berard
Department Name
Pediatric oncology
Contact Person Name
Nadege CORRADINI
Contact Person Email
nadege.corradini@ihope.fr

Sponsor

Primary sponsor

Full Name
F. Hoffmann-La Roche AG
Organisation Type
Pharmaceutical company
Country Of Registered Address
Switzerland

Contract research organisations

Name
IQVIA Limited
Responsibilities
sponsorDuties codes: [1]; contact eu_clinical_trials_information@iqvia.com
Name
Icon Development Solutions LLC
Responsibilities
sponsorDuties codes: [4]; sample management support (contact SampleManagementWhitesboro@iconplc.com)

Third parties

  • {"country":"United Kingdom","full_name":"IQVIA Limited","duties_or_roles":"sponsorDuties codes: [1]","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Labcorp Central Laboratory Services LP","duties_or_roles":"sponsorDuties codes: [4]","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Labcorp Early Development Laboratories Inc.","duties_or_roles":"sponsorDuties codes: [4]","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Signant Health Global LLC","duties_or_roles":"sponsorDuties codes: [3]","organisation_type":"Pharmaceutical company"}
  • {"country":"France","full_name":"Median Technologies","duties_or_roles":"sponsorDuties codes: [4]","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Caris Mpi Inc.","duties_or_roles":"Patient Recruitment/Retention Service Provider (sponsorDuties code 15)","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Icon Development Solutions LLC","duties_or_roles":"sponsorDuties codes: [4]","organisation_type":"Pharmaceutical company"}
  • {"country":"Switzerland","full_name":"Labcorp Central Laboratory Services SARL","duties_or_roles":"sponsorDuties codes: [4]","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Foundation Medicine Inc.","duties_or_roles":"sponsorDuties codes: [4]","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Greenphire LLC","duties_or_roles":"Patient Recruitment/Retention Service Provider (sponsorDuties code 15)","organisation_type":"Non-Pharmaceutical company"}
  • {"country":"Germany","full_name":"Foundation Medicine GmbH","duties_or_roles":"sponsorDuties codes: [4]","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Ventana Medical Systems Inc.","duties_or_roles":"sponsorDuties codes: [4]","organisation_type":"Pharmaceutical company"}
  • {"country":"Belgium","full_name":"CellCarta","duties_or_roles":"sponsorDuties codes: [4]","organisation_type":"Laboratory/Research/Testing facility"}

Investigational products

Investigational Product Name
INAVOLISIB
Active Substance
INAVOLISIB
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Maximum Dose
9 mg
Investigational Product Name
RO 743-5846/F04
Active Substance
DIVARASIB
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Investigational Product Name
RO7223619
Active Substance
BELVARAFENIB
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Maximum Dose
800 mg
Investigational Product Name
Ipatasertib
Active Substance
IPATASERTIB
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Maximum Dose
400 mg
Investigational Product Name
Rozlytrek 200 mg hard capsules
Active Substance
ENTRECTINIB
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Authorisation Status
Marketing authorisation (EU) (EU/1/20/1460/002)
Maximum Dose
600 mg
Investigational Product Name
Alecensa 150 mg hard capsules
Active Substance
ALECTINIB
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Authorisation Status
Marketing authorisation (IS) (EU/1/16/1169/001)
Maximum Dose
1200 mg
Investigational Product Name
Rozlytrek 100 mg hard capsules
Active Substance
ENTRECTINIB
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Authorisation Status
Marketing authorisation (EU) (EU/1/20/1460/001)
Maximum Dose
600 mg
Investigational Product Name
Tecentriq 1 200 mg concentrate for solution for infusion
Active Substance
ATEZOLIZUMAB
Modality
Monoclonal antibody
Routes Of Administration
IV INFUSION
Route
IV INFUSION
Authorisation Status
Marketing authorisation (EU) (EU/1/17/1220/001)
Maximum Dose
1200 mg
Investigational Product Name
Camonsertib
Active Substance
CAMONSERTIB
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Investigational Product Name
RO 749-9790/F02-02
Active Substance
PRALSETINIB
Modality
Small molecule
Routes Of Administration
ORAL
Route
ORAL
Maximum Dose
400 mg

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