Clinical trial • Phase II • Oncology
(3R)-N-[3-[5-(2-CYCLOPROPYLPYRIMIDIN-5-YL)-1H-PYRROLO[2,3-B]PYRIDINE-3-CARBONYL]-2,4-DIFLUOROPHENYL]-3-FLUOROPYRROLIDINE-1-SULFONAMIDE for Tumors harboring BRAF alterations | Primary central nervous system tumours with BRAF V600E mutation or BRAF fusions
Phase II trial of (3R)-N-[3-[5-(2-CYCLOPROPYLPYRIMIDIN-5-YL)-1H-PYRROLO[2,3-B]PYRIDINE-3-CARBONYL]-2,4-DIFLUOROPHENYL]-3-FLUOROPYRROLIDINE-1-SULFONAMIDE f…
Overview
- Trial Therapeutic Area
- Oncology
- Trial Disease
- Tumors harboring BRAF alterations | Primary central nervous system tumours with BRAF V600E mutation or BRAF fusions
- Trial Stage
- Phase II
- Drug Modality
- Small molecule
- Paediatric Trial
- Yes
Key dates
- Initial CTIS Submission Date
- 23-07-2024
- First CTIS Authorization Date
- 22-08-2024
Trial design
open-label, none/not specified-controlled Phase II trial in Spain, Italy, France and others.
- Open Label
- Yes
- Comparator
- None/Not specified
- Biomarker Stratified
- True: biomarker BRAF alterations (V600E mutation and BRAF fusions); strata by subprotocol (A: BRAF fusions; B: primary CNS tumors; C: rare BRAF V600E-mutated solid tumours; D: BRAF V600E solid tumours not eligible for other subprotocols)
- Target Sample Size
- 125
Eligibility
Recruits 125 paediatric patients.
- Vulnerable Population
- Vulnerable populations include pediatric participants (min age ≥10 years for subprotocols A, B, C; 16 years for subprotocol D). The submission includes age-specific assent and consent documents (assent forms for ages 8-11, 10-11, 12-16, 17 years; parent/guardian consent forms). Consent is obtained from adult participants; for minors, parent(s)/legal guardian(s) provide consent and age-appropriate assent is obtained from the minor. Multiple language ICF/assent templates are provided (country-specific).
Inclusion criteria
- {"criterion_text":"- Subprotocol A: 1. Male and female, ≥10 years of age, and weighing ≥30 kg.\n- Subprotocol C: 4. Have an archival tissue sample available meeting protocol requirements. If an archival tissue sample is not available, a newly obtained (before treatment) tumor biopsy may be submitted instead.\n- Subprotocol C: 5. Consent to provide scan(s) prior to baseline to assess change in tumor trajectory.\n- Subprotocol B: 3.Documented BRAF V600E mutation in tumor and/or blood detected by an analytically validated test at CLIA or CLIA-equivalent laboratory approved by sponsor or sponsor-designated central test.\n- Subprotocol C: 6. Received all available standard therapy, is intolerant to available therapies, or treatment with standard therapy is not appropriate.\n- Subprotocol D: 1. Male and female, 16-65 years of age.\n- Subprotocol D: 2. Histologic diagnosis of a solid tumor harboring a BRAFV600E mutation and not elegible for other subprotocols.\n- Subprotocol D: 3. Measurable disease on CT, MRI or physical exam\n- Subprotocol D: 4. Evidence of BRAF V600E mutation in tumor and/or blood detected by genomic tests\n- Subprotocol B: 4. An archival tissue sample available meeting protocol requirements, or fresh biopsy is required if the archival sample is not available for retrospective confirmation test. Tissue obtained most proximal to initiating this subprotocol is preferred.\n- Subprotocol B: 5. Measurable disease based upon specified response criteria, as determined by the radiographic BICR.\n- Subprotocol A: 5. Consent to provide scan(s) prior to baseline to assess change in tumor trajectory.\n- Subprotocol B: 6. All adverse events related to prior therapies (eg, chemotherapy, radiotherapy, surgery) must have resolved to Grade 1 or baseline except for: a. Alopecia (Grade ≤2) b. Sensory neuropathy (Grade ≤2) c. Other adverse events that have resolved to Grade ≤2 that, according to the clinical judgment of the investigator, do not constitute a safety risk to the participant\n- Subprotocol B: 7. Participants who are receiving corticosteroid treatment must be on a stable or decreasing dose of ≤8 mg/day of dexamethasone or equivalent corticosteroid treatment for 7 days prior to first dose of study treatments.\n- Subprotocol A: 2. Histologic diagnosis of a solid tumor or primary CNS tumor.\n- Subprotocol A: 3. Documentation of BRAF gene fusion in tumor and/or blood detected by an analytically validated test by DNA sequencing or RNA (transcriptome) sequencing at CLIA or CLIA-equivalent laboratory or sponsor-designated central laboratory.\n- Subprotocol A: 4. Have an archival tissue sample available meeting protocol requirements. If an archival tissue sample is not available, a newly obtained (before treatment) tumor biopsy may be submitted instead.\n- Subprotocol D: 5. Consent to provide a tumor biopsy.\n- Subprotocol D: 6. Willingness to comply with the ECG substudy procedures\n- Subprotocol D: 7. All AEs related to prior therapies must have resolved to grade 1 or baseline.\n- Subprotocol A: 6. Received all available standard therapy, is intolerant to available therapies, or the investigator has determined that treatment with standard therapy is not appropriate.\n- Subprotocol A: 7. All adverse events related to prior therapies (chemotherapy; radiotherapy; surgery) must have resolved to Grade 1 or baseline\n- Subprotocol B: 1. Male and female, ≥10 years of age, and weighing ≥30 kg.\n- Subprotocol B: 2. Histological diagnosis of a primary CNS tumor, including but not limited to the following: a. Adults (≥18 years) with Grade 1-4 glioma or glioneuronal tumor (including glioblastoma, anaplastic astrocytoma, high grade astrocytoma with piloid features, pilocytic astrocytoma, gliosarcoma, anaplastic pleomorphic xanthoastrocytoma, anaplastic oligodendroglioma, anaplastic oligoastrocytoma, not otherwise specified [NOS], ganglioglioma, or recurrent LGG), OR b. Pediatric patients (10-17 years of age) with a Grade 3 or 4 glioma or glioneuronal tumor, including those with a prior, histologically confirmed, diagnosis of a low-grade glioma or glioneuronal tumor and now have radiographic or histopathological findings consistent with WHO [2021] Grade 3 or 4 primary CNS tumor. c. Participants must have unresectable, locally advanced or metastatic disease that: i. Had prior treatment with radiotherapy and/or first-line chemotherapy or concurrent chemoradiation therapy (Note: Participants who have a WHO Grade 3 or 4 glioma for whom chemotherapy and/or radiotherapy is not considered standard of care may remain eligible for the study. Consult the Medical Lead to discuss and determine if participant is eligible for enrollment). OR ii. Is intolerant to available therapies OR iii. Treatment with standard therapy is not appropriate.\n- Subprotocol C: 1. Male and female, ≥10 years of age, and weighing ≥30 kg.\n- Subprotocol C: 2. Histologic diagnosis of a rare BRAF V600E-mutated solid tumor that is unresectable, locally advanced or metastatic.\n- Subprotocol C: 3. Documented BRAF V600E mutation in tumor and/or blood detected by an analytically validated test at CLIA or CLIA-equivalent laboratory approved by sponsor or sponsor-designated central test."}
Exclusion criteria
- {"criterion_text":"- Subprotocol A:3. Prior treatment with MAPK inhibitors active for Class 2 BRAF alterations for advanced unresectable or metastatic disease (including but not limited to tovorafenib [formerly known as DAY 101, TAK 580, and MLN 2480], KIN-2787, BGB-3245, andCFT1946). Note: Participants with pediatric-type LGGs (molecular classification byWHO2021; diagnosed at ≤25 years of age) who had received prior treatment(s)with RAF/BRAF inhibitors are eligible for enrollment, provided there was no evidence of tumor progression on that therapy or within 4 weeks of discontinuation, based upon radiographic assessment.\n- Subprotocol D: 2. Participant has CNS metastases.\n- Subprotocol B: 2. Known or suspected neurofibromatosis-1 (NF-1) and/or Ras related gene alterations.\n- Subprotocol A: 4. Tyrosine kinase inhibitor(s) and/or targeted therapies are allowed (other than BRAF/MAPK pathway inhibitors per Exclusion Criteria 3 and 4) and will be restricted to no more than the number of lines of therapy that are consistent with standard treatment guidelines. NOTE: There is no restriction on the number of lines of chemotherapy or immunotherapy.\n- Subprotocol D: 3. Uncontrolled intercurrent illness that would limit compliance with study requirements.\n- Subprotocol D: 4. Active infection requiring systemic therapy.\n- Subprotocol D: 5. Current or planned participation in a study of an investigational agent or device.\n- Subprotocol D: 6. Have impairment of gastrointestinal (GI) function or GI disease that may significantly alter the absorption of oral plixorafenib or cobicistat (such as ulcerative diseases, uncontrolled nausea, vomiting, diarrhea, malabsorption syndrome, small bowel resection).\n- Subprotocol D: 7. Grade ≥ 2 changes in AST, ALT, gamma-glutamyl transaminase (GGT), or bilirubin attributed to prior immune checkpoint inhibitor treatment are exclusionary, even if resolved.\n- Subprotocol D: 8. Use or anticipate the need for medications with known risk for QT-prolonging potential and Torsades de Pointes.\n- Subprotocol B: 3. Uncontrolled intercurrent illness that would limit compliance with study requirements.\n- Subprotocol C: 3. Participant has CNS metastases.\n- Subprotocol B: 4. Active infection requiring systemic therapy.\n- Subprotocol B: 5. Current or planned participation in a study of an investigational agent or device.\n- Subprotocol B: 6. Have impairment of gastrointestinal (GI) function or GI disease that may significantly alter the absorption of oral plixorafenib (such as ulcerative diseases, uncontrolled nausea, vomiting, diarrhea, malabsorption syndrome, small bowel resection).\n- Subprotocol A: 5. Malignancy with co-occurring activating RAS mutation(s) at any time.\n- Subprotocol B: 7. Grade ≥ 2 changes in AST, ALT, gamma-glutamyl transaminase (GGT), or bilirubin attributed to prior immune checkpoint inhibitor treatment are exclusionary, even if resolved.\n- Subprotocol D: 9. History of acute or chronic cardiovascular disease or surgery, hypertension, with systolic blood pressure > 160 mm Hg, history of QTc abnormalities, or clinical significant ECG abnormalities.\n- Subprotocol A: 6. Uncontrolled intercurrent illness that would limit compliance with study requirements.\n- Subprotocol A: 7. Current or planned participation in a study of an investigational agent or device.\n- Subprotocol A: 8. Have impairment of gastrointestinal (GI) function or GI disease that may significantly alter the absorption of oral plixorafenib (such as ulcerative diseases, uncontrolled nausea, vomiting, diarrhea, malabsorption syndrome, and small bowel resection).\n- Subprotocol C: 1. Diagnosis of colorectal adenocarcinoma or pancreatic ductal adenocarcinoma (neuroendocrine or acinar tumors are eligible).\n- Subprotocol C: 5. Known or suspected neurofibromatosis-1 (NF-1) and/or RAS related gene alterations.\n- Subprotocol C: 2. Diagnosis of BRAF V600E mutated melanoma, papillary thyroid cancer or NSCLC.\n- Subprotocol B: 1. Prior treatment with BRAF, ERK, and/or MEK inhibitor(s).\n- Subprotocol C: 4. Prior treatment with BRAF, ERK, and/or MEK inhibitor(s), unless otherwise specified for specific tumor types (i.e. low grade serios or borderline ovarian cancer)\n- Subprotocol C: 6. Uncontrolled intercurrent illness that would limit compliance with study requirements.\n- Subprotocol C: 7. Active infection requiring systemic therapy.\n- Subprotocol C: 8. Current or planned participation in a study of an investigational agent or device.\n- Subprotocol C: 9. Have impairment of gastrointestinal (GI) function or GI disease that may significantly alter the absorption of oral plixorafenib or cobicistat (such as ulcerative diseases, uncontrolled nausea, vomiting, diarrhea, malabsorption syndrome, small bowel resection).\n- Subprotocol C: 10. Grade ≥ 2 changes in AST, ALT, gamma-glutamyl transaminase (GGT), or bilirubin attributed to prior immune checkpoint inhibitor treatment are exclusionary, even if resolved.\n- Subprotocol D: 1. Known or suspected neurofibromatosis-1 (NF-1) and/or RAS related gene alterations."}
Endpoints
Primary endpoints
- {"endpoint_text":"- 1. Objective Response Rate (ORR) (Subprotocol A, B and C): ORR will be determined by standard tumor response criteria by blinded independent central review (BICR)","definition_or_measurement_approach":"ORR will be determined by standard tumor response criteria by blinded independent central review (BICR)."}
- {"endpoint_text":"- 2. Pharmacokinetics (Subprotocol D): Systemic exposure of plixorafenib measured by Cmax and AUC.","definition_or_measurement_approach":"Systemic exposure of plixorafenib measured by Cmax and AUC."}
Recruitment
- Digital Remote Recruitment
- True: digital methods described include Google Ads, landing pages and online patient materials (documented in recruitment materials, particularly for Spain).
- Planned Sample Size
- 125
- Recruitment Window Months
- 59
- Consent Approach
- Informed consent is obtained from adult participants. For minors, parent(s)/legal guardian(s) provide consent and age-appropriate assent is obtained (assent forms provided for multiple pediatric age bands including 8-11, 10-11, 12-16, 17). Consent and assent materials are provided in country-specific languages (examples: Italian, German, French, Spanish, Swedish, Norwegian, Dutch) and include specific pregnancy and prescreening documents as well as vendor consent (e.g. Greenphire payment information).
Methods
- Physician referral letters / HCP brochures (country-specific physician referral letters provided e.g. K2_* Physician Referral Letter documents).
- Patient brochures and HCP clinical trial brochures (country-specific, e.g. K2_NL Patient Brochure, K2_FR HCP brochure, K2_IT patient materials).
- Patient navigator scripts and landing pages (digital outreach) — Spain materials include Google Ad, Landing Page, Patient Navigator Script.
- Online advertising (Google Ad) and dedicated landing page (documented for Spain).
- Site-led recruitment via participating hospitals/oncology centres and phase I units (country-specific recruitment procedures K1_* documents).
Geography
- Total Number Of Sites
- 26
- Total Number Of Participants
- 134
Spain
- Earliest CTIS Part Ii Submission Date
- 13-08-2024
- Latest Decision Or Authorization Date
- 22-08-2024
- Processing Time Days
- 9
- Number Of Sites
- 6
- Number Of Participants
- 40
Sites
- Site Name
- Hospital Universitari Vall D Hebron
- Department Name
- Medical Oncology department
- Principal Investigator Name
- María Vieito Villar
- Principal Investigator Email
- mvieito@vhio.net
- Contact Person Name
- María Vieito Villar
- Contact Person Email
- mvieito@vhio.net
- Site Name
- University Hospital Virgen Del Rocio S.L.
- Department Name
- Phase I Unit
- Principal Investigator Name
- Alejandro Falcon Gonzalez
- Principal Investigator Email
- Alejandro.falcon.sspa@juntadeandalucia.es
- Contact Person Name
- Alejandro Falcon Gonzalez
- Contact Person Email
- Alejandro.falcon.sspa@juntadeandalucia.es
- Site Name
- Hospital Infantil Universitario Nino Jesus
- Department Name
- Pediatric HematologyOncology Department
- Principal Investigator Name
- Alvaro Lassaletta Atienza
- Principal Investigator Email
- alvaro.lassaletta@salud.madrid.org
- Contact Person Name
- Alvaro Lassaletta Atienza
- Contact Person Email
- alvaro.lassaletta@salud.madrid.org
- Site Name
- Hospital Universitario 12 De Octubre
- Department Name
- Medical Oncology department
- Principal Investigator Name
- Guillermo De Velasco Oria de Ruerda
- Principal Investigator Email
- gdvelasco.gdv@gmail.com
- Contact Person Name
- Guillermo De Velasco Oria de Ruerda
- Contact Person Email
- gdvelasco.gdv@gmail.com
- Site Name
- Hospital Clinico Universitario De Valencia
- Department Name
- Phase I and Precision Medicine Unit
- Principal Investigator Name
- Valentina Gambardella
- Principal Investigator Email
- VGambardella@incliva.es
- Contact Person Name
- Valentina Gambardella
- Contact Person Email
- VGambardella@incliva.es
- Site Name
- Complexo Hospitalario Universitario De Santiago
- Department Name
- Medical Oncology department
- Principal Investigator Name
- Alexandra Cortegoso
- Principal Investigator Email
- alexandra.sabela.cortegoso.mosquera@sergas.es
- Contact Person Name
- Alexandra Cortegoso
- Contact Person Email
- alexandra.sabela.cortegoso.mosquera@sergas.es
Italy
- Earliest CTIS Part Ii Submission Date
- 13-08-2024
- Latest Decision Or Authorization Date
- 17-09-2024
- Processing Time Days
- 35
- Number Of Sites
- 4
- Number Of Participants
- 8
Sites
- Site Name
- IRCCS Istituto Nazionale Tumori Fondazione Pascale
- Department Name
- Dipartimento Ematologia e Terapie Innovative
- Principal Investigator Name
- Paolo Ascierto
- Principal Investigator Email
- paolo.ascierto@gmail.com
- Contact Person Name
- Paolo Ascierto
- Contact Person Email
- paolo.ascierto@gmail.com
- Site Name
- Istituto Romagnolo Per Lo Studio Dei Tumori Dino Amadori IRST S.r.l.
- Department Name
- Oncourology
- Principal Investigator Name
- Alberto Farolfi
- Principal Investigator Email
- alberto.farolfi@irst.emr.it
- Contact Person Name
- Alberto Farolfi
- Contact Person Email
- alberto.farolfi@irst.emr.it
- Site Name
- Ospedale San Raffaele S.r.l.
- Department Name
- Unità di Oncologia Medica
- Principal Investigator Name
- Andrea Necchi
- Principal Investigator Email
- Necchi.andrea@hsr.it
- Contact Person Name
- Andrea Necchi
- Contact Person Email
- Necchi.andrea@hsr.it
- Site Name
- Istituto Europeo Di Oncologia S.r.l.
- Department Name
- Oncologia ed New Drug Development Division for Innovative Therapies
- Principal Investigator Name
- Giuseppe Curiliano
- Principal Investigator Email
- giuseppe.curigliano@ieo.it
- Contact Person Name
- Giuseppe Curiliano
- Contact Person Email
- giuseppe.curigliano@ieo.it
France
- Earliest CTIS Part Ii Submission Date
- 13-08-2024
- Latest Decision Or Authorization Date
- 03-09-2024
- Processing Time Days
- 21
- Number Of Sites
- 8
- Number Of Participants
- 40
Sites
- Site Name
- Centre Hospitalier Regional Et Universitaire De Brest
- Department Name
- Service Pneumologie
- Principal Investigator Name
- Jean-Philippe Metges
- Principal Investigator Email
- jean-philippe.metges@chu-brest.fr
- Contact Person Name
- Jean-Philippe Metges
- Contact Person Email
- jean-philippe.metges@chu-brest.fr
- Site Name
- Oncopole Claudius Regaud
- Department Name
- Unité de recherche Clinique
- Principal Investigator Name
- Delphine Larrieu
- Principal Investigator Email
- larrieur.delphine@iuct-oncopole.fr
- Contact Person Name
- Delphine Larrieu
- Contact Person Email
- larrieur.delphine@iuct-oncopole.fr
- Site Name
- Institut Gustave Roussy
- Department Name
- Service Oncologie Médicale
- Principal Investigator Name
- Samuel Abbou
- Principal Investigator Email
- samuel.abbou@gustaveroussy.fr
- Contact Person Name
- Samuel Abbou
- Contact Person Email
- samuel.abbou@gustaveroussy.fr
- Site Name
- Timone University Hospital
- Department Name
- Service d'Oncologie Multidisciplinaire et Innovations Thérapeutiques
- Principal Investigator Name
- Pascale Tomasini
- Principal Investigator Email
- pascale.tomasini@ap-hm.fr
- Contact Person Name
- Pascale Tomasini
- Contact Person Email
- pascale.tomasini@ap-hm.fr
- Site Name
- Institut De Cancerologie De L Ouest
- Department Name
- Service Oncologie Médicale
- Principal Investigator Name
- Pierre Kubicek
- Principal Investigator Email
- pierre.kubicek@ico.unicancer.fr
- Contact Person Name
- Pierre Kubicek
- Contact Person Email
- pierre.kubicek@ico.unicancer.fr
- Site Name
- Institut Bergonie
- Department Name
- Service Oncologie Médicale
- Principal Investigator Name
- Florent Peyraud
- Principal Investigator Email
- f.peyraud@bordeaux.unicancer.fr
- Contact Person Name
- Florent Peyraud
- Contact Person Email
- f.peyraud@bordeaux.unicancer.fr
- Site Name
- Hopitaux Universitaires Pitie Salpetriere
- Department Name
- Service Neurologie
- Principal Investigator Name
- Mehdi Touat
- Principal Investigator Email
- mehdi.touat@aphp.fr
- Contact Person Name
- Mehdi Touat
- Contact Person Email
- mehdi.touat@aphp.fr
- Site Name
- Institut De Cancerologie De L Ouest (additional listed site)
- Department Name
- Service Oncologie Médicale (duplicate listing across entries)
- Principal Investigator Name
- Pierre Kubicek
- Principal Investigator Email
- pierre.kubicek@ico.unicancer.fr
- Contact Person Name
- Pierre Kubicek
- Contact Person Email
- pierre.kubicek@ico.unicancer.fr
Germany
- Earliest CTIS Part Ii Submission Date
- 13-08-2024
- Latest Decision Or Authorization Date
- 30-08-2024
- Processing Time Days
- 17
- Number Of Sites
- 3
- Number Of Participants
- 16
Sites
- Site Name
- Krankenhaus Nordwest GmbH
- Department Name
- Institut für Klinisch-Onkologische Forschung (IKF)
- Principal Investigator Name
- Thorsten Oliver Götze
- Principal Investigator Email
- goetze.thorsten@khnw.de
- Contact Person Name
- Thorsten Oliver Götze
- Contact Person Email
- goetze.thorsten@khnw.de
- Site Name
- Universitaetsklinikum Heidelberg AöR
- Department Name
- Neurologische Klinik Neuroonkologie
- Principal Investigator Name
- Antje Wick
- Principal Investigator Email
- antje.wick@med.uni-heidelberg.de
- Contact Person Name
- Antje Wick
- Contact Person Email
- antje.wick@med.uni-heidelberg.de
- Site Name
- Charite Universitaetsmedizin Berlin KöR
- Department Name
- Medizinische Klinik mit Schwerpunkt Hämatologie, Onkologie und Tumorimmunologie (CVK)
- Principal Investigator Name
- Dominik Modest
- Principal Investigator Email
- dominik.modest@charite.de
- Contact Person Name
- Dominik Modest
- Contact Person Email
- dominik.modest@charite.de
Sweden
- Earliest CTIS Part Ii Submission Date
- 13-08-2024
- Latest Decision Or Authorization Date
- 23-08-2024
- Processing Time Days
- 10
- Number Of Sites
- 2
- Number Of Participants
- 15
Sites
- Site Name
- Region Skane Skanes Universitetssjukhus
- Department Name
- Department of Hematology, Oncology and Radiation Physics, SUS – Lund, Lasarettsg. 23 A, 221 85 Lund
- Principal Investigator Name
- Ana Carneiro
- Principal Investigator Email
- ana.carneiro@med.lu.se
- Contact Person Name
- Ana Carneiro
- Contact Person Email
- ana.carneiro@med.lu.se
- Site Name
- Karolinska University Hospital
- Department Name
- Department of Clinical Cancer Studies
- Principal Investigator Name
- Jeffrey Yachnin
- Principal Investigator Email
- jeffrey.yachnin@regionstockholm.se
- Contact Person Name
- Jeffrey Yachnin
- Contact Person Email
- jeffrey.yachnin@regionstockholm.se
Norway
- Earliest CTIS Part Ii Submission Date
- 21-04-2025
- Latest Decision Or Authorization Date
- 14-05-2025
- Processing Time Days
- 23
- Number Of Sites
- 2
- Number Of Participants
- 10
Sites
- Site Name
- Helse Bergen HF
- Department Name
- The Cancer Clinic
- Principal Investigator Name
- Kjersti Elvestad Hestetun
- Principal Investigator Email
- kjse@ihelse.net
- Contact Person Name
- Kjersti Elvestad Hestetun
- Contact Person Email
- kjse@ihelse.net
- Site Name
- Oslo University Hospital HF
- Department Name
- Oncology department
- Principal Investigator Name
- Tormod Kyrre Guren
- Principal Investigator Email
- uxtour@ous-hf.no
- Contact Person Name
- Tormod Kyrre Guren
- Contact Person Email
- uxtour@ous-hf.no
Netherlands
- Earliest CTIS Part Ii Submission Date
- 30-03-2026
- Latest Decision Or Authorization Date
- 24-04-2026
- Processing Time Days
- 25
- Number Of Sites
- 1
- Number Of Participants
- 5
Sites
- Site Name
- Erasmus Universitair Medisch Centrum Rotterdam (Erasmus MC)
- Department Name
- Internal Oncology
- Principal Investigator Name
- Marjolein Geurts
- Principal Investigator Email
- neuro-onco-trials@erasmusmc.nl
- Contact Person Name
- Marjolein Geurts
- Contact Person Email
- neuro-onco-trials@erasmusmc.nl
Sponsor
Primary sponsor
- Full Name
- Fore Biotherapeutics Inc.
- Organisation Type
- Pharmaceutical company
- Country Of Registered Address
- United States
Contract research organisations
- Name
- PPD Development LP
- Responsibilities
- PK samples
- Name
- Icon Clinical Research Limited
- Responsibilities
- PK samples; Tissue sample; Programming; DMC; MM; CTL; CT transparency; Legal rep
- Name
- Imaging Endpoints II LLC
- Responsibilities
- Medical image analysis/ review - X-ray, MRI, ultrasound, imaging or cat scan.
Third parties
- {"country":"United States","full_name":"Greenphire LLC","duties_or_roles":"Patient reimbursement","organisation_type":"Non-Pharmaceutical company"}
- {"country":"United States","full_name":"Tempus Labs Inc.","duties_or_roles":"NGS Testing","organisation_type":"Non-Pharmaceutical company"}
- {"country":"United States","full_name":"PPD Development LP","duties_or_roles":"PK samples","organisation_type":"Pharmaceutical company"}
- {"country":"Ireland","full_name":"Icon Clinical Research Limited","duties_or_roles":"PK samples; Tissue sample; Programming; DMC; MM; CTL; CT transparency; Legal rep","organisation_type":"Pharmaceutical company"}
- {"country":"United States","full_name":"Imaging Endpoints II LLC","duties_or_roles":"Medical image analysis/ review - X-ray, MRI, ultrasound, imaging or cat scan.","organisation_type":"Pharmaceutical company"}
- {"country":"United States","full_name":"Guardant Health Inc.","duties_or_roles":"NGS Testing","organisation_type":"Laboratory/Research/Testing facility"}
- {"country":"United States","full_name":"Eresearchtechnology Inc.","duties_or_roles":"ECG sub-study","organisation_type":"Pharmaceutical company"}
- {"country":"United States","full_name":"Medidata Solutions Inc.","duties_or_roles":"","organisation_type":"Non-Pharmaceutical company"}
- {"country":"United States","full_name":"Suvoda LLC","duties_or_roles":"Interactive response technologies (IRT)","organisation_type":"Non-Pharmaceutical company"}
- {"country":"United States","full_name":"Scout Clinical","duties_or_roles":"Patient reimbursement","organisation_type":"Hospital/Clinic/Other health care facility"}
- {"country":"Ireland","full_name":"Millmount Healthcare Limited (DP Packaging and Labelling/ Batch Certification/EU Importer)","duties_or_roles":"DP Packaging and Labelling/ Batch Certification/EU Importer","organisation_type":"Pharmaceutical company"}
- {"country":"Ireland","full_name":"Millmount Healthcare Limited (Batch Certification/EU Importation Site)","duties_or_roles":"Batch Certification/EU Importation Site","organisation_type":"Pharmaceutical company"}
Investigational products
- Investigational Product Name
- FORE8394 (PLX8394)
- Active Substance
- (3R)-N-[3-[5-(2-CYCLOPROPYLPYRIMIDIN-5-YL)-1H-PYRROLO[2,3-B]PYRIDINE-3-CARBONYL]-2,4-DIFLUOROPHENYL]-3-FLUOROPYRROLIDINE-1-SULFONAMIDE
- Modality
- Small molecule
- Routes Of Administration
- ORAL USE
- Route
- Oral
- Authorisation Status
- Investigational (IMP11566/00001)
- Investigational Product Name
- Tybost 150 mg film-coated tablets (COBICISTAT)
- Active Substance
- COBICISTAT
- Modality
- Small molecule
- Routes Of Administration
- ORAL USE
- Route
- Oral
- Authorisation Status
- Authorised (marketing authorisation EU/1/13/872/002 listed for Tybost)
- Starting Dose
- 150 mg
- Dose Levels
- 150 mg
- Maximum Dose
- 150 mg
- Combination Treatment
- Yes
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