Clinical trial • Phase III • Psychiatry

1-[6-ETHYL-8-FLUORO-4-METHYL-3-(3-METHYL-1,2,4-OXADIAZOL-5-YL)QUINOLIN-2-YL]-N-(OXAN-4-YL)PIPERIDIN-4-AMINE for Major Depressive Disorder

Phase III trial of 1-[6-ETHYL-8-FLUORO-4-METHYL-3-(3-METHYL-1,2,4-OXADIAZOL-5-YL)QUINOLIN-2-YL]-N-(OXAN-4-YL)PIPERIDIN-4-AMINE for Major Depressive Disord…

Overview

Trial Therapeutic Area
Psychiatry
Trial Disease
Major Depressive Disorder
Trial Stage
Phase III
Drug Modality
Small molecule

Key dates

Initial CTIS Submission Date
15-03-2024
First CTIS Authorization Date
20-06-2024

Trial design

Randomised, nmra-335140 arm: participants will receive 80mg nmra-335140 qd; placebo arm: participants will receive identical placebo nmra-335140 qd (placebo identical to active to maintain blinding).-controlled Phase III trial in Finland, France, Sweden and others.

Randomised
Yes
Comparator
NMRA-335140 Arm: Participants will receive 80mg NMRA-335140 QD; Placebo Arm: Participants will receive identical placebo NMRA-335140 QD (placebo identical to active to maintain blinding).
Target Sample Size
205
Trial Duration For Participant
42

Eligibility

Recruits 205 The trial record indicates vulnerable populations are selected (populationOfTrialSubjects.isVulnerablePopulationSelected = true). Subject information and consent form documents include caregiver and minor/pregnant-partner versions (e.g., document titles such as 'L1_CZ_SIS-ICF_Caregiver_Czech_redacted', 'L1_DE_SIS-ICF_Minor Pregnant Partner_German', 'L1_DE_SIS-ICF_Adult Pregnant Partner_German'), indicating procedures for obtaining consent/assent and caregiver involvement where applicable. Adult participants provide informed consent; caregiver-consent/assent materials are available as indicated by the document titles..

Vulnerable Population
The trial record indicates vulnerable populations are selected (populationOfTrialSubjects.isVulnerablePopulationSelected = true). Subject information and consent form documents include caregiver and minor/pregnant-partner versions (e.g., document titles such as 'L1_CZ_SIS-ICF_Caregiver_Czech_redacted', 'L1_DE_SIS-ICF_Minor Pregnant Partner_German', 'L1_DE_SIS-ICF_Adult Pregnant Partner_German'), indicating procedures for obtaining consent/assent and caregiver involvement where applicable. Adult participants provide informed consent; caregiver-consent/assent materials are available as indicated by the document titles.

Inclusion criteria

  • {"criterion_text":"- Have a primary Diagnostic and Statistical Manual of Mental Disorders Fifth Edition Text Revised (DSM-5-TR) diagnosis of MDD without psychotic features confirmed by Structured Clinical Interview for DSM 5 Disorders, Clinical Trials Version (SCID 5 CT) at screening (this may be a first or recurrent episode)."}
  • {"criterion_text":"- Participant's current major depressive episode must be confirmed by independent assessment."}
  • {"criterion_text":"- The symptoms of the current MDD episode have been present for more than 4 weeks prior to the Screening Visit, but no longer than 12 months prior to the Screening Visit."}
  • {"criterion_text":"- Have a MADRS total score of 25 or higher at Screening and Baseline."}
  • {"criterion_text":"- A change in MADRS total score between Screening and Baseline of ≤20%."}

Exclusion criteria

  • {"criterion_text":"- Have failed 2 or more courses of antidepressant treatment at sufficient doses for at least 6 to 8 weeks for the current MDD episode."}
  • {"criterion_text":"- Currently or in the past year have been diagnosed with a personality disorder per the DSM-5-TR or in the past 3 years have been diagnosed with any of the following DSM-5-TR disorders: anorexia nervosa, bulimia nervosa, or binge eating disorder. Participants with comorbid generalized anxiety disorder, social anxiety disorder, simple phobias, or panic disorder for whom MDD is considered the primary diagnosis are not excluded."}
  • {"criterion_text":"- Have a lifetime diagnosis of bipolar 1 or 2, schizophrenia or schizoaffective, schizophreniform, obsessive compulsive disorder, or post-traumatic stress disorder (PTSD)."}
  • {"criterion_text":"- Have moderate to severe substance or alcohol use disorder, per DSM-5-TR criteria, within the 12 months prior to screening (excluding nicotine)."}
  • {"criterion_text":"- Are actively suicidal (eg, any suicide attempts within the past 12 months) or are at serious suicidal risk as indicated by any current suicidal intent, including a plan, as assessed by the Columbia Suicide Severity Rating Scale (C-SSRS) (score of \"YES\" on suicidal ideations Item 4 or 5 within 3 months prior to Visit 1 [Screening]) and/or based on clinical evaluation by the Investigator; or are homicidal, in the opinion of the Investigator. Participants who are currently hospitalized for MDD symptoms or suicidality are not allowed into the study. If there is a recent history (within 3 months of screening) of hospitalization due to MDD symptoms, the participant should be discussed with the Medical Monitor for eligibility."}

Endpoints

Primary endpoints

  • {"endpoint_text":"- The primary endpoint is the treatment difference in change from Baseline to Week 6 in the MADRS total score.","definition_or_measurement_approach":"Change from Baseline to Week 6 in the MADRS (Montgomery-Åsberg Depression Rating Scale) total score."}

Secondary endpoints

  • {"endpoint_text":"- Participant reported symptoms of anhedonia. Change from Baseline to Week 6 assessed in the Snaith-Hamilton Pleasure Scale (SHAPS) total score. Change from Baseline to each timepoint assessed in the SHAPS total score","definition_or_measurement_approach":"Change from Baseline to Week 6 and to each timepoint in SHAPS total score (Snaith-Hamilton Pleasure Scale)."}
  • {"endpoint_text":"- MADRS response rate. Percentage of participants whose MADRS total score decreased by greater than or equal to 50% from Baseline.","definition_or_measurement_approach":"Percentage of participants with ≥50% reduction in MADRS total score from Baseline."}
  • {"endpoint_text":"- MADRS scores over time. Change from Baseline to each timepoint assessed in MADRS total scores.","definition_or_measurement_approach":"Change from Baseline to each scheduled timepoint in MADRS total score."}
  • {"endpoint_text":"- Clinical assessment of MDD severity and improvement. Change from Baseline to each timepoint assessed in Clinical Global Impression of Severity (CGIS) score. Value at each timepoint assessed in Clinical Global Impression of Improvement (CGI-I) score","definition_or_measurement_approach":"Change from Baseline in CGI-S at each timepoint; CGI-I value at each timepoint."}
  • {"endpoint_text":"- Participant reported symptoms of MDD. Change from Baseline to each timepoint assessed in Patient Health Questionnaire9 (PHQ9) total score","definition_or_measurement_approach":"Change from Baseline to each timepoint in PHQ-9 total score."}
  • {"endpoint_text":"- Participant reported severity of anhedonia. Change from Baseline to each timepoint assessed in PHQ9 Anhedonia Item #1","definition_or_measurement_approach":"Change from Baseline to each timepoint in PHQ-9 item #1 (anhedonia)."}
  • {"endpoint_text":"- Clinician reported symptoms of anxiety. Change from Baseline to each timepoint assessed in the Hamilton Anxiety Rating Scale (HAMA) total score","definition_or_measurement_approach":"Change from Baseline to each timepoint in HAM-A total score."}
  • {"endpoint_text":"- Participant reported assessment of functional impairment. Change from Baseline at Week 6 assessed in the Sheehan Disability Scale (SDS) total score","definition_or_measurement_approach":"Change from Baseline to Week 6 in SDS total score."}
  • {"endpoint_text":"- MADRS remission rate. Percentage of participants whose MADRS total score decreased to 10 or less","definition_or_measurement_approach":"Percentage of participants with MADRS total score ≤10 at assessment (remission rate)."}

Recruitment

Registry Or Advocacy Recruitment
True, Autocruitment LLC (Patient organisation/association) and Ctsdatabase LLC (Clinical trial subject registry) are named third parties with recruitment/registry roles.
Digital Remote Recruitment
True, digital/remote methods explicitly referenced include website materials, digital advertising, Instagram ads, landing pages, and digital prescreening tools (documents: e.g., 'K2_*_Digital Materials_Bilingual', 'K2_*_Instagram Ads', 'K2_*_landingpage').
Planned Sample Size
205
Recruitment Window Months
10
Consent Approach
Informed consent is obtained using subject information and informed consent form documents. ICF and subject information documents are available in multiple country-specific languages as indicated by document titles (examples: Czech, German, Polish, Bulgarian, French, Swedish). There are specific caregiver and minor/pregnant-partner consent/assent documents (e.g., 'L1_CZ_SIS-ICF_Caregiver', 'L1_DE_SIS-ICF_Minor Pregnant Partner', 'L1_DE_SIS-ICF_Adult Pregnant Partner'), indicating age- or role-specific consent procedures and caregiver consent handling where applicable.

Methods

  • Website recruitment materials (country-specific website PDFs listed for Czech, Germany, Poland, Bulgaria).
  • Digital materials and Instagram ads (documents: 'K2_*_Digital Materials_Bilingual', 'K2_*_Instagram Ads').
  • Printed materials: Posters, Flyers, Brochures (documents: 'K2_*_Poster', 'K2_*_PDF Flyer', 'K2_*_Brochure').
  • Newspaper advertisements (documents: 'K2_*_Newspaper Ad' e.g., Czech/Polish/Bulgarian/German versions).
  • Display Ads / Web banners / Landing page (documents: 'K2_*_Display Ads', 'landingpage_Pratia sites_German').
  • Telephone recruitment scripts and prescreening tools (documents: 'Telephone Script_Bilingual', 'prescreening_tool_questions').
  • Scout / patient concierge and email outreach materials (documents: 'Scout Email', 'Scout Study Brochure').
  • Country-specific printed and digital recruitment campaigns (document titles include country codes CZ/DE/PL/BG and are tailored per country site lists).

Geography

Total Number Of Sites
34
Total Number Of Participants
127

Finland

Earliest CTIS Part Ii Submission Date
05-06-2024
Latest Decision Or Authorization Date
24-06-2024
Processing Time Days
19
Number Of Sites
3
Number Of Participants
9

Sites

Site Name
Clinical Research Services Turku CRST Oy
Contact Person Name
Noora Scheinin
Contact Person Email
nmsche@utu.fi
Site Name
Lahdelma Consulting Oy
Contact Person Name
Liisa Lahdelma
Contact Person Email
liisa.lahdelma@kolumbus.fi
Site Name
Oulu Mentalcare Oy
Contact Person Name
Markku Timonen
Contact Person Email
markku.timonen@mentalcare.fi

France

Earliest CTIS Part Ii Submission Date
11-06-2024
Latest Decision Or Authorization Date
28-06-2024
Processing Time Days
17
Number Of Sites
7
Number Of Participants
18

Sites

Site Name
University Hospital Of Clermont-Ferrand
Department Name
Département de Psychiatrie
Contact Person Name
Ludovic Samalin
Site Name
Desbonnet Recherche
Contact Person Name
Philippe Desbonnet
Site Name
Centre Hospitalier Henri Laborit
Department Name
Department of Psychiatry and Medical Psychology
Contact Person Name
Nematollah Jaafari
Contact Person Email
Nemat.jaafari@ch-poitiers.fr
Site Name
Centre Hospitalier Universitaire De Montpellier
Department Name
Service Universitaire de Psychiatrie Adulte
Contact Person Name
Jérôme Attal
Contact Person Email
j-attal@chu-montpellier.fr
Site Name
Centre Hospitalier Georges Mazurelle- EPSM Mazurelle
Department Name
Département de Psychiatrie
Contact Person Name
Anne Sauvaget
Contact Person Email
Anne.sauvaget@chu-nantes.fr
Site Name
Centre Hospitalier Universitaire De Nimes
Department Name
Pôle Psychiatrie
Contact Person Name
Fabrice Boulet
Contact Person Email
fabrice.boulet@chu-nimes.fr
Site Name
Centre Hospitalier Universitaire D'Angers
Department Name
Département de Psychiatrie
Contact Person Name
Bénédicte Gohier
Contact Person Email
begohier@chu-angers.fr

Sweden

Earliest CTIS Part Ii Submission Date
05-06-2024
Latest Decision Or Authorization Date
20-06-2024
Processing Time Days
15
Number Of Sites
2
Number Of Participants
6

Sites

Site Name
ProbarE i Stockholm AB (Lund location)
Department Name
ProbareE location in Lund
Contact Person Name
Anders Luts
Contact Person Email
anders.luts@probare.se
Site Name
ProbarE i Stockholm AB (Stockholm location)
Contact Person Name
Peter Bosson
Contact Person Email
peter.bosson@probare.se

Czechia

Earliest CTIS Part Ii Submission Date
25-06-2024
Latest Decision Or Authorization Date
08-07-2024
Processing Time Days
13
Number Of Sites
3
Number Of Participants
22

Sites

Site Name
INEP medical s.r.o.
Contact Person Name
Alexander Nawka
Contact Person Email
nawka@inep.cz
Site Name
Brain-Soultherapy s.r.o.
Contact Person Name
Claudia Vodičková-Borzová
Contact Person Email
cborzova@seznam.cz
Site Name
A-Shine s.r.o.
Department Name
Psychiatrie
Contact Person Name
Luboš Janů
Contact Person Email
lubos.janu@seznam.cz

Germany

Earliest CTIS Part Ii Submission Date
11-06-2024
Latest Decision Or Authorization Date
28-06-2024
Processing Time Days
17
Number Of Sites
5
Number Of Participants
11

Sites

Site Name
Charite Universitaetsmedizin Berlin KöR
Department Name
Department of Psychiatry and Neurosciences
Contact Person Name
Dimitris Repantis
Contact Person Email
dimitris.repantis@charite.de
Site Name
Nervenärztliche Praxis Frau Dr. Kirsten HahN
Department Name
Arztpraxis für Neurologie und Psychatrie
Contact Person Name
Kirsten Hahn
Contact Person Email
hahnkirsten@gmail.com
Site Name
Klinische Forschung Hamburg GmbH
Department Name
Neurologie und Psychiatrie
Contact Person Name
Christian Deckert
Contact Person Email
christian.deckert@pratia.com
Site Name
Klinische Forschung Berlin-Mitte GmbH
Department Name
-
Contact Person Name
Sameer Kulkarni
Contact Person Email
sameer.kulkarni@pratia.com
Site Name
Emovis GmbH
Department Name
Dedicated Study Site
Contact Person Name
Sascha Öhm
Contact Person Email
sascha.oehm@emovis.de

Poland

Earliest CTIS Part Ii Submission Date
25-06-2024
Latest Decision Or Authorization Date
05-07-2024
Processing Time Days
10
Number Of Sites
6
Number Of Participants
27

Sites

Site Name
Promente Sp. z o.o.
Contact Person Name
Katarzyna Łachut
Contact Person Email
rejestracja@pro-mente.pl
Site Name
E4r&D Sp. z o.o.
Contact Person Name
Wiesław J. Cubała
Contact Person Email
cubala@gumed.edu.pl
Site Name
Indywidualna Specjalistyczna Praktyka Lekarska Agnieszka Remlinger-Molenda
Contact Person Name
Agnieszka Remlinger-Molenda
Contact Person Email
aremlinger@gmail.com
Site Name
Ginemedica Sp. z o.o.
Contact Person Name
Ewa Tylko
Contact Person Email
e.tylko@ginemedica.pl
Site Name
Prywatne Gabinety Lekarskie 'Promedicus' Anna Agnieszka Tomczak
Contact Person Name
Anna Agnieszka Tomczak
Contact Person Email
promedicus@onet.eu
Site Name
Centrum Medyczne Luxmed Sp. z o.o.
Contact Person Name
Dariusz Malicki
Contact Person Email
dariuszmalicki@interia.eu

Bulgaria

Earliest CTIS Part Ii Submission Date
31-05-2024
Latest Decision Or Authorization Date
01-07-2024
Processing Time Days
31
Number Of Sites
8
Number Of Participants
34

Sites

Site Name
Diagnostic And Consultation Centre St.Vrach And St.St. Kuzma And Damian OOD
Department Name
Not applicable
Contact Person Name
Petya Dimitrova
Contact Person Email
drdimitrova@abv.bg
Site Name
Multiprofile Hospital For Active Treatment - Targovishte AD
Department Name
Department of Psychiatry
Contact Person Name
Ivan Tyanev
Contact Person Email
dr.ivan.tyanev@gmail.com
Site Name
Diagnostics-Consultancy Center Mladost M Varna OOD
Department Name
Not applicable
Contact Person Name
Hristo Kozhuharov
Contact Person Email
christokojuharov@abv.bg
Site Name
Medical Center Lifemed EOOD
Department Name
Not applicable
Contact Person Name
Rozaliya Rangelova
Contact Person Email
rrangelova80@gmail.com
Site Name
Dr. Ivo Natsov Outpatient Clinic For Individual Practice For Specialized Medical Care In Psychiatry ET
Department Name
Not applicable
Contact Person Name
Ivo Natsov
Contact Person Email
ivo_nacov@abv.bg
Site Name
Medical Center Intermedica Ltd.
Department Name
Not applicable
Contact Person Name
Toni Donchev
Contact Person Email
tonyd@abv.bg
Site Name
Medical Center Akademica EOOD
Department Name
Not applicable
Contact Person Name
Vihra Milanova
Contact Person Email
vihra.milanova@gmail.com
Site Name
Medical Center (additional listed site)
Department Name
Not applicable
Contact Person Name
Toni Donchev
Contact Person Email
tonyd@abv.bg

Sponsor

Primary sponsor

Full Name
Neumora Therapeutics Inc.
Organisation Type
Pharmaceutical company
Country Of Registered Address
United States

Contract research organisations

Name
Icon Clinical Research Limited
Responsibilities
Multiple sponsor duties listed (codes: 1,11,12,13,2,3,4,5,6,8) indicating broad CRO responsibilities as recorded in CTIS thirdParties.sponsorDuties
Name
Tigermed-Bdm Inc.
Responsibilities
Sponsor duties code: 10 (listed in CTIS thirdParties.sponsorDuties)
Name
WCG Clinical Inc.
Responsibilities
eCOA, Rater Training (sponsor duties codes: 13, 15 listed)
Name
Almac Clinical Services Limited
Responsibilities
Sponsor duties code: 14 (listed in CTIS thirdParties.sponsorDuties)

Third parties

  • {"country":"United States","full_name":"Mms Holdings Inc.","duties_or_roles":"Pharmacovigilance","organisation_type":"Pharmaceutical company"}
  • {"country":"Ireland","full_name":"Icon Clinical Research Limited","duties_or_roles":"Sponsor duties codes: 1,11,12,13,2,3,4,5,6,8 (as listed in CTIS thirdParties.sponsorDuties)","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Psomagen Inc.","duties_or_roles":"Sponsor duties codes: 13,4","organisation_type":"Laboratory/Research/Testing facility"}
  • {"country":"United States","full_name":"Massachusetts General Hospital","duties_or_roles":"Independent depression study eligibility assessment","organisation_type":"Hospital/Clinic/Other health care facility"}
  • {"country":"United States","full_name":"Tigermed-Bdm Inc.","duties_or_roles":"Sponsor duties codes: 10","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Alturas Analytics Inc.","duties_or_roles":"Sponsor duties codes: 13,4","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Medidata Solutions Inc.","duties_or_roles":"Sponsor duties codes: 7","organisation_type":"Non-Pharmaceutical company"}
  • {"country":"United States","full_name":"Eresearchtechnology Inc.","duties_or_roles":"Sponsor duties codes: 13 and 15 (Cardiac safety)","organisation_type":"Pharmaceutical company"}
  • {"country":"France","full_name":"Hydrogen","duties_or_roles":"recruitment","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"WCG Clinical Inc.","duties_or_roles":"Sponsor duties codes: 13 and 15 (eCOA, Rater Training)","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Aicure LLC","duties_or_roles":"IP compliance","organisation_type":"Non-Pharmaceutical company"}
  • {"country":"United States","full_name":"Autocruitment LLC","duties_or_roles":"Participant recruitment","organisation_type":"Patient organisation/association"}
  • {"country":"United States","full_name":"Ctsdatabase LLC","duties_or_roles":"Clinical trial subject registry","organisation_type":"Non-Pharmaceutical company"}
  • {"country":"United Kingdom (Northern Ireland)","full_name":"Almac Clinical Services Limited","duties_or_roles":"Sponsor duties codes: 14","organisation_type":"Pharmaceutical company"}
  • {"country":"United States","full_name":"Scout Clinical","duties_or_roles":"Patient concierge","organisation_type":"Hospital/Clinic/Other health care facility"}
  • {"country":"France","full_name":"Quipment","duties_or_roles":"Equipment - Konan Microscope","organisation_type":"Non-Pharmaceutical company"}
  • {"country":"United States","full_name":"Voiant","duties_or_roles":"Ophthalmology","organisation_type":"Health care"}

Investigational products

Investigational Product Name
NMRA-335140
Active Substance
1-[6-ETHYL-8-FLUORO-4-METHYL-3-(3-METHYL-1,2,4-OXADIAZOL-5-YL)QUINOLIN-2-YL]-N-(OXAN-4-YL)PIPERIDIN-4-AMINE
Modality
Small molecule
Routes Of Administration
ORAL
Route
Oral
Authorisation Status
Investigational (marketingAuthNumber: N/A; prodAuthStatus: 1 as recorded)
Starting Dose
80 mg
Dose Levels
80 mg
Frequency
QD
Maximum Dose
80 mg
Investigational Product Name
Placebo is identical to the active NMRA-335140 but without the active drug substance to maintain study blinding.
Modality
Other
Routes Of Administration
ORAL
Route
Oral
Frequency
QD

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